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- [1] Clinical activity of the mutant-selective EGFR inhibitor AZD9291 in patients with EGFR inhibitor-resistant non-small cell lung cancer[J]. TRANSLATIONAL LUNG CANCER RESEARCH, 2014, 3 (06) : 370 - 372Jiang, Tao论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ, Shanghai Pulm Hosp, Sch Med, Dept Oncol, Shanghai 200433, Peoples R China Tongji Univ, Shanghai Pulm Hosp, Sch Med, Dept Oncol, Shanghai 200433, Peoples R ChinaZhou, Caicun论文数: 0 引用数: 0 h-index: 0机构: Tongji Univ, Shanghai Pulm Hosp, Sch Med, Dept Oncol, Shanghai 200433, Peoples R China Tongji Univ, Shanghai Pulm Hosp, Sch Med, Dept Oncol, Shanghai 200433, Peoples R China
- [2] AZD9291 in EGFR Inhibitor-Resistant Non-Small-Cell Lung Cancer[J]. NEW ENGLAND JOURNAL OF MEDICINE, 2015, 372 (18): : 1689 - 1699Jaenne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USA Dana Farber Canc Inst, Belfer Inst Appl Canc Sci, Boston, MA 02215 USA Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAYang, James Chih-Hsin论文数: 0 引用数: 0 h-index: 0机构: Natl Taiwan Univ, Taipei 10764, Taiwan Natl Taiwan Univ Hosp, Taipei, Taiwan Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAKim, Dong-Wan论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ Hosp, Seoul 110744, South Korea Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAPlanchard, David论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, France Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAOhe, Yuichiro论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Tokyo, Japan Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USARamalingam, Suresh S.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USA Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAAhn, Myung-Ju论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ Hlth Syst, Samsung Med Ctr, Seoul, South Korea Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAKim, Sang-We论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ Hlth Syst, Asan Med Ctr, Seoul, South Korea Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USASu, Wu-Chou论文数: 0 引用数: 0 h-index: 0机构: Cheng Kung Univ Hosp, Taipei, Taiwan Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAHorn, Leora论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN USA Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAHaggstrom, Daniel论文数: 0 引用数: 0 h-index: 0机构: Carolinas Healthcare Syst, Levine Canc Inst, Charlotte, NC USA Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAFelip, Enriqueta论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Univ Hosp, Barcelona, Spain Vall dHebron Inst Oncol, Barcelona, Spain Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAKim, Joo-Hang论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ Hlth Syst, Yonsei Canc Ctr, Seoul, South Korea Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAFrewer, Paul论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield, Cheshire, England Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USACantarini, Mireille论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield, Cheshire, England Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USABrown, Kathryn H.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield, Cheshire, England Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USADickinson, Paul A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield, Cheshire, England Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USAGhiorghiu, Serban论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield, Cheshire, England Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USARanson, Malcolm论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Christie Hosp, Manchester, Lancs, England Dana Farber Canc Inst, Lowe Ctr Thorac Oncol, Boston, MA 02215 USA
- [3] AZD9291, a mutant-selective EGFR inhibitor, as first-line treatment for EGFR mutation-positive advanced non-small cell lung cancer (NSCLC): Results from a phase 1 expansion cohort.[J]. JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Ramalingam, Suresh S.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAYang, James Chih-Hsin论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USALee, Chee Khoon论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAKurata, Takayasu论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAKim, Dong-Wan论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAJohn, Thomas论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USANogami, Naoyuki论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAOhe, Yuichiro论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USARukazenkov, Yuri论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAFrewer, Paul论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USACantarini, Mireille论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAGhiorghiu, Serban论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USAJanne, Pasi A.论文数: 0 引用数: 0 h-index: 0机构: Emory Univ, Winship Canc Inst, Atlanta, GA 30322 USA
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- [5] Osimertinib (AZD9291), a Mutant-Selective EGFR Inhibitor, Reverses ABCB1-Mediated Drug Resistance in Cancer Cells[J]. MOLECULES, 2016, 21 (09)Zhang, Xiao-Yu论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAZhang, Yun-Kai论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAWang, Yi-Jun论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAGupta, Pranav论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAZeng, Leli论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA Sun Yat Sen Univ, Sch Chem & Chem Engn, Guangzhou 510275, Guangdong, Peoples R China St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAXu, Megan论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA John L Miller Great Neck North High Sch, Great Neck, NY 11023 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAWang, Xiu-Qi论文数: 0 引用数: 0 h-index: 0机构: South China Agr Univ, Coll Anim Sci, Guangzhou 510642, Guangdong, Peoples R China St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAYang, Dong-Hua论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USAChen, Zhe-Sheng论文数: 0 引用数: 0 h-index: 0机构: St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA St Johns Univ, Dept Pharmaceut Sci, Coll Pharm & Hlth Sci, Queens, NY 11439 USA
- [6] Osimertinib (AZD9291), a mutant-selective EGFR inhibitor, reverses ABCB1-mediated drug resistance in cancer cells[J]. CANCER RESEARCH, 2017, 77Zhang, Xiao-Yu论文数: 0 引用数: 0 h-index: 0Lei, Zi-Ning论文数: 0 引用数: 0 h-index: 0Zhang, Yun-Kai论文数: 0 引用数: 0 h-index: 0Wang, Yi-Jun论文数: 0 引用数: 0 h-index: 0Gupta, Pranav论文数: 0 引用数: 0 h-index: 0Zeng, Leli论文数: 0 引用数: 0 h-index: 0Xu, Megan论文数: 0 引用数: 0 h-index: 0Wang, Xiu-Qi论文数: 0 引用数: 0 h-index: 0Yang, Dong-Hua论文数: 0 引用数: 0 h-index: 0Chen, Zhe-Sheng论文数: 0 引用数: 0 h-index: 0
- [7] Acquired Resistance to the Mutant-Selective EGFR Inhibitor AZD9291 Is Associated with Increased Dependence on RAS Signaling in Preclinical Models[J]. CANCER RESEARCH, 2015, 75 (12) : 2489 - 2500Eberlein, Catherine A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandStetson, Daniel论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandMarkovets, Aleksandra A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandAl-Kadhimi, Katherine J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandLai, Zhongwu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandFisher, Paul R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield SK10 4TG, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandMeador, Catherine B.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Dept Med, Nashville, TN USA Vanderbilt Univ, Vanderbilt Ingram Canc Ctr, Nashville, TN 37235 USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandSpitzler, Paula论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Dept Med, Nashville, TN USA Vanderbilt Univ, Vanderbilt Ingram Canc Ctr, Nashville, TN 37235 USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandIchihara, Eiki论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Dept Med, Nashville, TN USA Vanderbilt Univ, Vanderbilt Ingram Canc Ctr, Nashville, TN 37235 USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandRoss, Sarah J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandAhdesmaki, Miika J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandAhmed, Ambar论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandRatcliffe, Laura E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield SK10 4TG, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandO'Brien, Elizabeth L. Christey论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield SK10 4TG, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandBarnes, Claire H.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandBrown, Henry论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandSmith, Paul D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandDry, Jonathan R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandBeran, Garry论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandThress, Kenneth S.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandDougherty, Brian论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Waltham, MA USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandPao, William论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Dept Med, Nashville, TN USA Vanderbilt Univ, Vanderbilt Ingram Canc Ctr, Nashville, TN 37235 USA AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, EnglandCross, Darren A. E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England AstraZeneca, Macclesfield SK10 4TG, Cheshire, England AstraZeneca Oncol Innovat Med, Macclesfield, Cheshire, England
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- [10] Loss of EGFR confers acquired resistance to AZD9291 in an EGFR-mutant non-small cell lung cancer cell line with an epithelial–mesenchymal transition phenotype[J]. Journal of Cancer Research and Clinical Oncology, 2018, 144 : 1413 - 1422Jing Xu论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalXiaoting Zhao论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalDengfeng He论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalJinghui Wang论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalWeiying Li论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalYinghui Liu论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalLi Ma论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalMei Jiang论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalYu Teng论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalZiyu Wang论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalMeng Gu论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalJianbin Wu论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalYue Wang论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalWentao Yue论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest HospitalShucai Zhang论文数: 0 引用数: 0 h-index: 0机构: Capital Medical University,Department of Medical Oncology, Beijing Tuberculosis and Thoracic Tumor Research Institute/Beijing Chest Hospital