INHIBITION OF EFS-, PHENYLEPHRINE-, AND THROMBOXANE-INDUCED CONTRACTION BY THE RECEPTOR ANTAGONIST, PICOTAMIDE, IN HUMAN PROSTATE SMOOTH MUSCLE

被引:0
|
作者
Hennenberg, Martin
Miljak, Marijan
Strittmatter, Frank
Hocaoglu, Yasemin
Rutz, Beata
Fuellhase, Claudius
Stief, Christian G.
Gratzke, Christian
机构
来源
JOURNAL OF UROLOGY | 2013年 / 189卷 / 04期
关键词
D O I
10.1016/j.juro.2013.02.3145
中图分类号
R5 [内科学]; R69 [泌尿科学(泌尿生殖系疾病)];
学科分类号
1002 ; 100201 ;
摘要
1595
引用
收藏
页码:E655 / E656
页数:2
相关论文
共 43 条
  • [1] The receptor antagonist picotamide inhibits adrenergic and thromboxane-induced contraction of hyperplastic human prostate smooth muscle
    Hennenberg, Martin
    Miljak, Marijan
    Herrmann, Daniel
    Strittmatter, Frank
    Walther, Sebastian
    Rutz, Beata
    Hocaoglu, Yasemin
    Kunit, Thomas
    Schreiber, Andrea
    Andersson, Karl-Erik
    Stief, Christian G.
    Gratzke, Christian
    AMERICAN JOURNAL OF PHYSIOLOGY-RENAL PHYSIOLOGY, 2013, 305 (10) : F1383 - F1390
  • [2] INHIBITION OF NEUROGENIC, CHOLINERGIC, AND ADRENERGIC CONTRACTION OF HUMAN BLADDER SMOOTH MUSCLE BY THE THROMBOXANE RECEPTOR ANTAGONIST, PICOTAMIDE
    Hennenberg, Martin
    Wang, Yiming
    Strittmatter, Frank
    Ciotkowska, Anna
    Rutz, Beata
    Stief, Christian
    Gratzke, Christian
    JOURNAL OF UROLOGY, 2016, 195 (04): : E891 - E892
  • [3] THE INHIBITION BY FPL-55712 OF THROMBOXANE-INDUCED BRONCHIAL SMOOTH-MUSCLE CONTRACTION INVIVO
    SMITH, GM
    MOTION, MC
    MALLARKEY, G
    INTERNATIONAL JOURNAL OF MICROCIRCULATION-CLINICAL AND EXPERIMENTAL, 1984, 3 (3-4): : 420 - 420
  • [4] Thromboxane-induced ERK phosphorylation in human aortic smooth muscle cells
    Gallet, C
    Blaie, S
    Lévy-Toledano, S
    Habib, A
    ADVANCES IN PROSTAGLANDIN, LEUKOTRIENE, AND OTHER BIOACTIVE LIPID RESEARCH: BASIC SCIENCE AND CLINICAL APPLICATIONS, 2003, 525 : 71 - 73
  • [5] EFFECTS OF THE RECEPTOR ANTAGONIST PICOTAMIDE ON ENDOTHELIN-1-,-2-AND-3-INDUCED CONTRACTIONS IN HUMAN PROSTATE SMOOTH MUSCLE
    Tamalunas, Alexander
    Gratzke, Christian
    Strittmatter, Frank
    Waidelich, Raphaela
    Stief, Christian
    Hennenberg, Martin
    JOURNAL OF UROLOGY, 2016, 195 (04): : E603 - E604
  • [6] Inhibition of agonist-induced smooth muscle contraction by picotamide in the male human lower urinary tract outflow region
    Hennenberg, Martin
    Tamalunas, Alexander
    Wang, Yiming
    Keller, Patrick
    Schott, Melanie
    Strittmatter, Frank
    Herlemann, Annika
    Yu, Qingfeng
    Rutz, Beata
    Ciotkowska, Anna
    Stief, Christian G.
    Gratzke, Christian
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2017, 803 : 39 - 47
  • [7] Propofol potentiates phenylephrine-induced contraction via cyclooxygenase inhibition in pulmonary artery smooth muscle
    Ogawa, K
    Tanaka, S
    Murray, PA
    ANESTHESIOLOGY, 2001, 94 (05) : 833 - 839
  • [8] Inhibition of human prostate stromal cell growth and smooth muscle contraction by thalidomide: A novel remedy in LUTS?
    Tamalunas, Alexander
    Sauckel, Cora
    Ciotkowska, Anna
    Rutz, Beata
    Wang, Ruixiao
    Huang, Ru
    Li, Bingsheng
    Stief, Christian G.
    Gratzke, Christian
    Hennenberg, Martin
    PROSTATE, 2021, 81 (07): : 377 - 389
  • [9] Identification of a dihydropyridine as a potent α1a adrenoceptor-selective antagonist that inhibits phenylephrine-induced contraction of the human prostate
    Wong, WC
    Chiu, G
    Wetzel, JM
    Marzabadi, MR
    Nagarathnam, D
    Wang, D
    Fang, J
    Miao, SW
    Hong, XF
    Forray, C
    Vaysse, PJJ
    Branchek, TA
    Gluchowski, C
    Tang, R
    Lepor, H
    JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (14) : 2643 - 2650
  • [10] Thromboxane A2 induces contraction of human prostate smooth muscle by Rho kinase- and calmodulin-dependent mechanisms
    Strittmatter, Frank
    Gratzke, Christian
    Weinhold, Philipp
    Steib, Christian J.
    Hartmann, Anna C.
    Schlenker, Boris
    Andersson, Karl-Erik
    Hedlund, Petter
    Stief, Christian G.
    Hennenberg, Martin
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2011, 650 (2-3) : 650 - 655