共 50 条
- [1] Transcriptional Antagonism by CDK8 Inhibition Improves Therapeutic Efficacy of MEK InhibitorsCANCER RESEARCH, 2023, 83 (02) : 285 - 300Malone, Clare F.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Broad Inst MIT & Harvard, Cambridge, MA USA Harvard Med Sch, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAKim, Minjee论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Broad Inst MIT & Harvard, Cambridge, MA USA Harvard Med Sch, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAAlexe, Gabriela论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Broad Inst MIT & Harvard, Cambridge, MA USA Harvard Med Sch, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAEngel, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Broad Inst MIT & Harvard, Cambridge, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAForman, Alexandra B.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Broad Inst MIT & Harvard, Cambridge, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USARobichaud, Amanda论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA AstraZeneca, Waltham, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAConway, Amy Saur论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAGoodale, Amy论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAMeyer, Ashleigh论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAKhalid, Delan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAThayakumar, Allen论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAHatcher, John M.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Stanford Univ, Dept Chem & Syst Biol, ChEM H, Stanford, CA USA Stanford Univ, Stanford Canc Inst, Stanford, CA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAPiccioni, Federica论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA USA Merck Res Labs, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USAStegmaier, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA Broad Inst MIT & Harvard, Cambridge, MA USA Harvard Med Sch, Boston, MA USA Boston Childrens Hosp, Div Hematol Oncol, Boston, MA USA Dana Farber Canc Inst, Dept Pediat Oncol, Boston, MA USA
- [2] CDK8 as a therapeutic target for cancers and recent developments in discovery of CDK8 inhibitorsEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 164 : 77 - 91Xi, Meiyang论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaChen, Tingkai论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Jiangsu, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaWu, Chunlei论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaGao, Xiaozhong论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaWu, Yonghua论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaLuo, Xiang论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaDu, Kui论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaYu, Lemao论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaCai, Tao论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaShen, Runpu论文数: 0 引用数: 0 h-index: 0机构: Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R ChinaSun, Haopeng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Jiangsu, Peoples R China Shaoxing Univ, Coll Chem & Chem Engn, Shaoxing 312000, Peoples R China
- [3] Preventing adaptive therapeutic resistance to CDK4/6 inhibition with CDK8/19 inhibitorsCANCER RESEARCH, 2022, 82 (04)Mack, Zachary论文数: 0 引用数: 0 h-index: 0Yastrebova, Margarita论文数: 0 引用数: 0 h-index: 0Khamidullina, Alvina论文数: 0 引用数: 0 h-index: 0Sharko, Amanda论文数: 0 引用数: 0 h-index: 0Ding, Xiaokai论文数: 0 引用数: 0 h-index: 0Bowe, Stephan论文数: 0 引用数: 0 h-index: 0Sashi, Nikitha论文数: 0 引用数: 0 h-index: 0Safa, Samantha论文数: 0 引用数: 0 h-index: 0Digsby, Kaitlyn论文数: 0 引用数: 0 h-index: 0Eckstrom, Amanda论文数: 0 引用数: 0 h-index: 0Sikirzhitski, Vitali论文数: 0 引用数: 0 h-index: 0Lim, Chang-Uk论文数: 0 引用数: 0 h-index: 0Tatarskiy, Victor论文数: 0 引用数: 0 h-index: 0Roninson, Igor论文数: 0 引用数: 0 h-index: 0Broude, Eugenia论文数: 0 引用数: 0 h-index: 0
- [4] CDK8/CDK19 inhibition as therapeutic target of metastatic prostate cancerVIRCHOWS ARCHIV, 2017, 471 : S269 - S269Offermann, A.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyBecker, F.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyKluemper, N.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyVogel, W.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyBraegelmann, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, GermanyPerner, S.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp UKSH, Inst Pathol, Lubeck, Germany Univ Hosp UKSH, Inst Pathol, Lubeck, Germany
- [5] CDK8 Inhibitors Induce Transcriptional Reprogramming of AML Cells Associated with DifferentiationBLOOD, 2019, 134Mazan, Milena论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandChapellier, Marion论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Div Clin Genet, Dept Lab Med, Lund, Sweden Selvita SA, Krakow, PolandJaras, Marcus论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Div Clin Genet, Dept Lab Med, Lund, Sweden Selvita SA, Krakow, PolandMikula, Michal论文数: 0 引用数: 0 h-index: 0机构: Maria Sklodowska Curie Mem Canc Ctr & Inst Oncol, Dept Genet, Warsaw, Poland Selvita SA, Krakow, PolandMajewska, Eliza论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandWiklik, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandCombik, Michal论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandGolas, Aniela论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandMasiejczyk, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandFiedor, Elzbieta论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandMalusa, Federico论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandJuszczynski, Przemyslaw论文数: 0 引用数: 0 h-index: 0机构: Inst Hematol & Transfus Med, Dept Expt Hematol, Warsaw, Poland Selvita SA, Krakow, PolandCybulska, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Maria Sklodowska Curie Mem Canc Ctr & Inst Oncol, Dept Genet, Warsaw, Poland Selvita SA, Krakow, PolandMikulski, Maciej论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandOstrowski, Jerzy论文数: 0 引用数: 0 h-index: 0机构: Maria Sklodowska Curie Mem Canc Ctr & Inst Oncol, Dept Genet, Warsaw, Poland Selvita SA, Krakow, PolandChrom, Pawel论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandBrzozka, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, PolandRzymski, Tomasz论文数: 0 引用数: 0 h-index: 0机构: Selvita SA, Krakow, Poland Selvita SA, Krakow, Poland
- [6] CDK8 inhibition improves the efficacy of ER- and HER2-targeted drugs in breast cancerCANCER RESEARCH, 2017, 77McDermott, M. S.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USAChumanevich, A.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USALiang, J.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USAChen, M.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USAAltilia, S.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USAHennes, C.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USARoninson, I. B.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USABroude, E. V.论文数: 0 引用数: 0 h-index: 0机构: Univ South Carolina, Columbia, SC 29208 USA Univ South Carolina, Columbia, SC 29208 USA
- [7] Taking Aim at Glycolysis with CDK8 InhibitorsTRENDS IN ENDOCRINOLOGY AND METABOLISM, 2018, 29 (05): : 281 - 282Fisher, Robert P.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Oncol Sci, New York, NY 10029 USA
- [8] In Search of Novel CDK8 Inhibitors by Virtual ScreeningJOURNAL OF CHEMICAL INFORMATION AND MODELING, 2017, 57 (03) : 413 - 416Kumarasiri, Malika论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaTeo, Theodosia论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaYu, Mingfeng论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaPhilip, Stephen论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaBasnet, Sunita K. C.论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaAlbrecht, Hugo论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaSykes, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaWang, Peng论文数: 0 引用数: 0 h-index: 0机构: Yabao Pharmaceut Grp Co Ltd, Suzhou Ind Pk, Suzhou 215123, Peoples R China Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, AustraliaWang, Shudong论文数: 0 引用数: 0 h-index: 0机构: Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia Univ South Australia, Sch Pharm & Med Sci, Adelaide, SA 5001, Australia Univ South Australia, Ctr Drug Discovery & Dev, Ctr Canc Biol, Sansom Inst Hlth Res, Adelaide, SA 5001, Australia
- [9] Biomarker Discovery for Cancer Sensitivity to CDK8 InhibitorsFASEB JOURNAL, 2018, 32 (01):Lu, Zhixin论文数: 0 引用数: 0 h-index: 0Spear, Jensen E.论文数: 0 引用数: 0 h-index: 0Russu, Wade A.论文数: 0 引用数: 0 h-index: 0
- [10] CDK8/19 inhibitors: 3-benzylindazolesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Schiemann, Kai论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyMallinger, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Merck Serono, Merck KGaA, Darmstadt, GermanyWienke, Dirk论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyEsdar, Christina论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyPoeschke, Oliver论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyBusch, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyRohdich, Felix论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyEccles, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Merck Serono, Merck KGaA, Darmstadt, GermanySchneider, Richard论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyRaynaud, Florence论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Merck Serono, Merck KGaA, Darmstadt, GermanyCzodrowski, Paul论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyMusil, Djordje论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanySchwarz, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyUrbahns, Klaus论文数: 0 引用数: 0 h-index: 0机构: Merck Serono, Merck KGaA, Darmstadt, Germany Merck Serono, Merck KGaA, Darmstadt, GermanyBlagg, Julian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, London, England Merck Serono, Merck KGaA, Darmstadt, Germany