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- [1] Potent anti-tumor activity of AUR102, a selective covalent inhibitor of CDK7EUROPEAN JOURNAL OF CANCER, 2020, 138 : S47 - S47Satyam, L. K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaPoddutoori, R.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Med Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaThiyagarajan, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaMukherjee, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Computat Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaKaza, L. N.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaCharamanna, K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Toxicol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaMarappan, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Biochem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaSamiulla, D.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaTiwari, N. K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaDevaraja, T.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Med Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaAravind, A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Pharmacol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaDhudashiya, A. A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaBooher, R.论文数: 0 引用数: 0 h-index: 0机构: Exelixis Inc, Alameda, CA USA Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaDaginakatte, G.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Pharmacol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaAntony, T.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Biochem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaChelur, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Toxicol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaNellore, K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaGiri, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaRamachandra, M.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaSamajdar, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Med Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India
- [2] SY-5609, an orally available selective CDK7 inhibitor demonstrates broad anti-tumor activity in vivoCANCER RESEARCH, 2019, 79 (13)Hu, Shanhu论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMarineau, Jason论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAHamman, Kristin论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USABradley, Michael论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USASavinainen, Anneli论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAAlnemy, Sydney论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USARajagopal, Nisha论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOrlando, David论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAChuaqui, Claudio论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOlson, Eric论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USA
- [3] An oral and selective CDK7 inhibitor demonstrates substantial anti-tumor effect in breast and ovarian cancer modelsEUROPEAN JOURNAL OF CANCER, 2018, 103 : E39 - E40Hu, S.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USAMarineau, J.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USABradley, M.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USAHamman, K.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USAAlnemy, S.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USASmith, D.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USACarulli, J.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USAChuaqui, C.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA Syros Pharmaceut Inc, Drug Discovery, Cambridge, MA USA
- [4] SY-1365, a potent and selective CDK7 inhibitor, exhibits promising anti-tumor activity in multiple preclinical models of aggressive solid tumorsCANCER RESEARCH, 2017, 77Hu, Shanhu论文数: 0 引用数: 0 h-index: 0Ke, Nan论文数: 0 引用数: 0 h-index: 0Ren, Yixuan论文数: 0 引用数: 0 h-index: 0Miljovska, Sofija论文数: 0 引用数: 0 h-index: 0Rajagopal, Nisha论文数: 0 引用数: 0 h-index: 0McKeown, Michael论文数: 0 引用数: 0 h-index: 0Orlando, David论文数: 0 引用数: 0 h-index: 0Sprott, Kevin论文数: 0 引用数: 0 h-index: 0Choi, Yoon J.论文数: 0 引用数: 0 h-index: 0Olson, Eric论文数: 0 引用数: 0 h-index: 0Fritz, Christian C.论文数: 0 引用数: 0 h-index: 0
- [5] Synergistic Anti-Tumor Effect of Combining Selective CDK7 and BRD4 Inhibition in NeuroblastomaFRONTIERS IN ONCOLOGY, 2022, 11Gao, Yang论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA Boston Childrens Hosp, Boston, MA 02115 USA Harvard Med Sch, Dept Pediat, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Nasholm, Nicole论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Pediat, San Francisco, CA 94143 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USADas, Sanjukta论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA Boston Childrens Hosp, Boston, MA 02115 USA Harvard Med Sch, Dept Pediat, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAKwiatkowski, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAAbraham, Brian J.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Computat Biol, 332 N Lauderdale St, Memphis, TN 38105 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAZhang, Tinghu论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAGustafson, Clay论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Pediat, San Francisco, CA 94143 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:George, Rani E.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA Boston Childrens Hosp, Boston, MA 02115 USA Harvard Med Sch, Dept Pediat, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA
- [6] Olomoucine derived synthetic CDK inhibitors: Selective induction of apoptotic death in tumor cells and in vivo anti-tumor activity are mediated via direct inhibition of cdk7ANNALS OF ONCOLOGY, 1998, 9 : 136 - 136Hajduch, M论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicNoskova, V论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicHavlieek, L论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicFeketova, G论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicGojova, L论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicKrystof, V论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicVesely, J论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicStrnad, M论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech RepublicMihal, V论文数: 0 引用数: 0 h-index: 0机构: Palacky Univ, Fac Med, CR-77520 Olomouc, Czech Republic
- [7] Q901; a highly selective covalent cdk7 inhibitor inducing substantial anti-tumor effect in a broad spectrum of solid tumor lineagesCANCER RESEARCH, 2022, 82 (12)Yu, Donghoon论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaJeon, Yeejin论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaLee, Seung-Joo论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaKim, Jaeseung论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaNam, Kiyean论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South Korea
- [8] Functional dissection of CDK7 in transcription using a highly selective CDK7 inhibitor Q901CANCER RESEARCH, 2024, 84 (06)Jung, Hyerim论文数: 0 引用数: 0 h-index: 0Um, Dahun论文数: 0 引用数: 0 h-index: 0Lee, Yoonji论文数: 0 引用数: 0 h-index: 0Yu, Donghoon论文数: 0 引用数: 0 h-index: 0Lee, Dayoung论文数: 0 引用数: 0 h-index: 0Ahn, Jiye论文数: 0 引用数: 0 h-index: 0Kim, Jeongjun论文数: 0 引用数: 0 h-index: 0Lee, Seung-Joo论文数: 0 引用数: 0 h-index: 0Kim, Jaeseung论文数: 0 引用数: 0 h-index: 0Nam, Kiyean论文数: 0 引用数: 0 h-index: 0Kim, Tae-Kyung论文数: 0 引用数: 0 h-index: 0
- [9] An oral and selective CDK12 inhibitor demonstrates robust anti-tumor activity.CANCER RESEARCH, 2022, 82 (12)Hu, Shanhu论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMoebius, David论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USADworakowski, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USACooper, Elliott论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USALaPlaca, Derek论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAAlnemy, Sydney论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAPerera, Phone论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMarineau, Jason论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAChuaqui, Claudio论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USACarulli, John P.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOlson, Eric论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USA
- [10] Development of TGN-1076, a selective and reversible small molecule inhibitor of CDK7CANCER RESEARCH, 2020, 80 (16)Thode, Trason论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USALi, Zhaoliang论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USAWeston, Alexis论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USADana, Srikanta论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USAAmpanattu, Sherin Daniel论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USASoldi, Raffaella论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USAKaadige, Mohan Rao论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USAVankayalapti, Hariprasad论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USAChung, Vincent论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, Duarte, CA USA TGen Translat Genom Res Inst, Phoenix, AZ USAChao, Joseph论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, Duarte, CA USA TGen Translat Genom Res Inst, Phoenix, AZ USAVon Hoff, Daniel D.论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USASharma, Sunil论文数: 0 引用数: 0 h-index: 0机构: TGen Translat Genom Res Inst, Phoenix, AZ USA TGen Translat Genom Res Inst, Phoenix, AZ USA