Evaluation of a Novel P-glycoprotein Inducer Using [18F] MC225 and PET

被引:0
|
作者
Varela, L. Garcia [1 ]
Garcia, D. Vallez [1 ]
Perez Rodriguez, M. [2 ]
Moraga-Amaro, R. [1 ]
Colabufo, N. A. [3 ]
Aguiar, P. [4 ]
Sobrino, T. [2 ]
Dierckx, R. A. J. O. [1 ]
van Waarde, A. [1 ]
Elsinga, P. H. [1 ]
Luurtsema, G. [1 ]
机构
[1] Univ Groningen, Univ Med Ctr Groningen, Dept Nucl Med & Mol Imaging, Groningen, Netherlands
[2] IDIS Hlth Res Inst, Clin Neurosci Res Lab, Santiago De Compostela, Spain
[3] Univ Bari Aldo Moro, Dept Pharm, Bari, Italy
[4] Clin Univ Hosp, IDIS Hlth Res Inst, Dept Nucl Med & Mol Imaging, Santiago De Compostela, Spain
关键词
TRANSPORTERS; BRAIN;
D O I
暂无
中图分类号
R8 [特种医学]; R445 [影像诊断学];
学科分类号
1002 ; 100207 ; 1009 ;
摘要
OP-221
引用
收藏
页码:S113 / S113
页数:1
相关论文
共 50 条
  • [1] In Vivo Induction of P-Glycoprotein Function can be Measured with [18F]MC225 and PET
    Garcia-Varela, Lara
    Rodriguez-Perez, Manuel
    Custodia, Antia
    Moraga-Amaro, Rodrigo
    Colabufo, Nicola A.
    Aguiar, Pablo
    Sobrino, Tomas
    Dierckx, Rudi A. J. O.
    van Waarde, Aren
    Elsinga, Philip H.
    Luurtsema, Gert
    MOLECULAR PHARMACEUTICS, 2021, 18 (08) : 3073 - 3085
  • [2] Quantification of P-glycoprotein function at the human blood-brain barrier using [18F]MC225 and PET
    Mossel, P.
    Willemsen, A. T.
    Varela, L. Garcia
    Arif, W.
    Boellaard, R.
    Elsinga, P. H.
    de Deyn, P.
    Dierckx, R. A.
    Lammertsma, A. A.
    Bartels, A. L.
    Luurtsema, G.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2021, 48 (SUPPL 1) : S295 - S296
  • [3] Quantification of P-glycoprotein function at the human blood-brain barrier using [18F]MC225 and PET
    Mossel, Pascalle
    Arif, Wejdan M.
    De Souza, Giordana Salvi
    Varela, Lara Garcia
    van der Weijden, Chris W. J.
    Boersma, Hendrikus H.
    Willemsen, Antoon T. M.
    Boellaard, Ronald
    Elsinga, Philip H.
    Borra, Ronald J. H.
    Dierckx, Rudi A. J. O.
    Lammertsma, Adriaan A.
    Bartels, Anna L.
    Luurtsema, Gert
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2023, 50 (13) : 3917 - 3927
  • [4] Quantification of P-glycoprotein function at the human blood-brain barrier using [18F]MC225 and PET
    Pascalle Mossel
    Wejdan M. Arif
    Giordana Salvi De Souza
    Lara Garcia Varela
    Chris W. J. van der Weijden
    Hendrikus H. Boersma
    Antoon T. M. Willemsen
    Ronald Boellaard
    Philip H. Elsinga
    Ronald J. H. Borra
    Rudi A. J. O. Dierckx
    Adriaan A. Lammertsma
    Anna L. Bartels
    Gert Luurtsema
    European Journal of Nuclear Medicine and Molecular Imaging, 2023, 50 : 3917 - 3927
  • [5] Dose-response assessment of cerebral P-glycoprotein inhibition in vivo with [18F]MC225 and PET
    Garcia-Varela, Lara
    Mossel, Pascalle
    Aguiar, Pablo
    Vazquez-Matias, Daniel A.
    van Waarde, Aren
    Willemsen, Antoon T. M.
    Bartels, Anna L.
    Colabufo, Nicola A.
    Dierckx, Rudi A. J. O.
    Elsinga, Philip H.
    Luurtsema, Gert
    JOURNAL OF CONTROLLED RELEASE, 2022, 347 : 500 - 507
  • [6] Oral Administration of [18F]MC225 for Quantification of P-glycoprotein Function: A Feasibility Study
    de Souza, Giordana Salvi
    Furini, Cristiane R. G.
    Sijbesma, Juergen W. A.
    Kominia, Maria
    Doorduin, Janine
    Giacobbo, Bruno Lima
    Lammertsma, Adriaan A.
    Tsoumpas, Charalampos
    Luurtsema, Gert
    MOLECULAR IMAGING AND BIOLOGY, 2025, 27 (01) : 89 - 98
  • [7] Pre-Clinical Assessment of Cardiac P-glycoprotein Function In Vivo with [18F]MC225 PET Imaging
    Liu, W.
    Mossel, P.
    Sijbesma, J.
    Doorduin, J.
    Dannenberg, M.
    Schwach, V.
    Slart, R. H. J. A.
    Luurtsema, G.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2024, 51 : S439 - S439
  • [8] Evaluation of P-glycoprotein function at the blood–brain barrier using [18F]MC225-PET
    Pascalle Mossel
    Lara Garcia Varela
    Wejdan M. Arif
    Chris W. J. van der Weijden
    Hendrikus H. Boersma
    Antoon T. M. Willemsen
    Ronald Boellaard
    Philip H. Elsinga
    Ronald J. H. Borra
    Nicola A. Colabufo
    Jun Toyohara
    Peter Paul de Deyn
    Rudi A. J. O. Dierckx
    Adriaan A. Lammertsma
    Anna L. Bartels
    Gert Luurtsema
    European Journal of Nuclear Medicine and Molecular Imaging, 2021, 48 : 4105 - 4106
  • [9] Blood-brain barrier P-glycoprotein function in Alzheimer's disease measured with [18F]MC225 and PET
    Mossel, P.
    da Souza, G. Salvi
    Willemsen, A. T. M.
    Somsen, J. F.
    Stormezand, G. N.
    de Deyn, P.
    Dierckx, R. A. J. O.
    Lammertsma, A. A.
    Verwey, N. A.
    Reesink, F.
    Bartels, A. L.
    Luurtsema, G.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2024, 51 : S265 - S265
  • [10] Test-retest variability of measuring P-glycoprotein function at the blood-brain barrier using [18F]MC225 and PET
    Mossel, P.
    de Souza, G. Salvi
    Willemsen, A. T. M.
    Elsinga, P. H.
    de Deyn, P.
    Dierckx, R. A. J.
    Lammertsma, A. A.
    Bartels, A. L.
    Luurtsema, G.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2022, 49 (SUPPL 1) : S557 - S558