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- [1] Design, synthesis and evaluation of potent DNA-alkylating agents for use in antibody-drug conjugates (ADCs)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 254Reid, Emily论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAArcher, Katie论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USABai, Chen论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAYoder, Nicholas论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAVitharana, Dilrukshi论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USALanieri, Leanne论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USABogalhas, Megan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAWu, Rui论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAQu, Qifeng论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAMaloney, Erin论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAAb, Olga论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAPonte, Jose论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAChari, Ravi论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAMiller, Michael论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USA
- [2] Design, synthesis, and evaluation of a novel class of potent DNA-alkylating agents for use in antibody-drug conjugates (ADCs)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247Li, Wei论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAReid, Emily论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAArcher, Katie论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAFishkin, Nathan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USADandeneau, Andre论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAKovtun, Yelena论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAHarvey, Lauren论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAWhiteman, Kathy论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAMiller, Michael L.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USAChari, Ravi论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen INC, Waltham, MA 02451 USA ImmunoGen INC, Waltham, MA 02451 USA
- [3] Design, synthesis, and evaluation of a novel class of potent DNA-alkylating agents for use in antibody-drug conjugates (ADCs)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250Miller, Michael论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USA
- [4] Design, synthesis and evaluation of novel, potent DNA alkylating agents and their antibody-drug conjugates (ADCs)BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (17) : 2455 - 2458Reid, Emily E.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAArcher, Katie E.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAShizuka, Manami论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAMcShea, Molly A.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAMaloney, Erin K.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAAb, Olga论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USALanieri, Leanne论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAWilhelm, Alan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAPonte, Jose F.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAYoder, Nicholas C.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAChari, Ravi V. J.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAMiller, Michael L.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA
- [5] Antibody-drug conjugates (ADCs) of indolino-benzodiazepine DNA-alkylating agentsCANCER RESEARCH, 2015, 75Miller, Michael L.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAShizuka, Manami论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAFishkin, Nathan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAReid, Emily论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAArcher, Katie论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAMaloney, Erin论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USABai, Chen论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAAb, Olga论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAYoder, Nick C.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAWu, Rui论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAHong, Erica论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USABogalhas, Megan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAWilhelm, Alan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAWhiteman, Kathleen论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAChari, Ravi论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USA
- [6] New class of DNA-alkylating agents with a suitable tolerability profile created for use in antibody-drug conjugates (ADCs).MOLECULAR CANCER THERAPEUTICS, 2013, 12 (11)Miller, Michael论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAFishkin, Nathan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USALi, Wei论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAReid, Emily论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAArcher, Katie论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAMaloney, Erin论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAKovtun, Yelena论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAJones, Gregory论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAEllis, Megan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USASingh, Rajeeva论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAWhiteman, Kathleen论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAPinkas, Jan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAChari, Ravi论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USA
- [7] Peptide-linked indolino-benzodiazepine DNA-alkylating agents for use in antibody-drug conjugates (ADCs)CANCER RESEARCH, 2016, 76Shizuka, Manami论文数: 0 引用数: 0 h-index: 0Wilhelm, Alan论文数: 0 引用数: 0 h-index: 0Archer, Katie论文数: 0 引用数: 0 h-index: 0Reid, Emily论文数: 0 引用数: 0 h-index: 0Yoder, Nicholas C.论文数: 0 引用数: 0 h-index: 0Bai, Chen论文数: 0 引用数: 0 h-index: 0Fishkin, Nathan论文数: 0 引用数: 0 h-index: 0Harris, Luke论文数: 0 引用数: 0 h-index: 0Maloney, Erin论文数: 0 引用数: 0 h-index: 0Hong, Erica论文数: 0 引用数: 0 h-index: 0Wu, Rui论文数: 0 引用数: 0 h-index: 0Ab, Olga论文数: 0 引用数: 0 h-index: 0Lai, Kate论文数: 0 引用数: 0 h-index: 0Sikka, Surina论文数: 0 引用数: 0 h-index: 0Jin, Shan论文数: 0 引用数: 0 h-index: 0Pinkas, Jan论文数: 0 引用数: 0 h-index: 0Chari, Ravi论文数: 0 引用数: 0 h-index: 0Miller, Michael L.论文数: 0 引用数: 0 h-index: 0
- [8] Synthesis of Highly Potent N-10 Amino-Linked DNA-Alkylating Indolinobenzodiazepine Antibody-Drug Conjugates (ADCs)ACS MEDICINAL CHEMISTRY LETTERS, 2019, 10 (08): : 1211 - 1215Archer, Katie E.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAReid, Emily E.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAShizuka, Manami论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA Pharmaron Inc, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAWoods, James论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA Alkermes Inc, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAHarris, Luke论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAMaloney, Erin K.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USABartle, Laura M.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAAb, Olga论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAWilhelm, Alan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USASetiady, Yulius论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAPonte, Jose F.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USASingh, Rajeeva论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAKeating, Thomas A.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAChari, Ravi V. J.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USAMiller, Michael L.论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA ImmunoGen Inc, 830 Winter St, Waltham, MA 02451 USA
- [9] Design and synthesis of potent DNA alkylating indolino-benzodiazepine compounds (BIAs) linked with a DNA binding moiety for use in antibody-drug conjugates (ADCs)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256Reid, Emily论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAArcher, Katie论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAShizuka, Manami论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAMcShea, Molly论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAMaloney, Erin论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAAb, Olga论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USALanieri, Leanne论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAWilhelm, Alan论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAPonte, Jose论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAYoder, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAChari, Ravi论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USAMiller, Michael论文数: 0 引用数: 0 h-index: 0机构: Immunogen Inc, Waltham, MA USA Immunogen Inc, Waltham, MA USA
- [10] Antibody-Drug Conjugates (ADCs) with novel IGN DNA-alkylating agents display potent antigen-specific activity against hematologic and solid tumor xenograft models.MOLECULAR CANCER THERAPEUTICS, 2013, 12 (11)Whiteman, Kathleen论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAJohnson, Holly论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAWilhelm, Alan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAMiller, Michael论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USALi, Wei论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAReid, Emily论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAArcher, Katie论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAFishkin, Nathan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USADandeneau, Andre论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAMaloney, Erin论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAPinkas, Jan论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USAChari, Ravi论文数: 0 引用数: 0 h-index: 0机构: ImmunoGen Inc, Waltham, MA USA ImmunoGen Inc, Waltham, MA USA