共 37 条
- [1] Bromodomain inhibitor OTX015 (MK-8628) combined with targeted agents shows strong in vivo antitumor activity in lymphoma[J]. ONCOTARGET, 2016, 7 (36) : 58142 - 58147Gaudio, Eugenio论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandTarantelli, Chiara论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandPonzoni, Maurilio论文数: 0 引用数: 0 h-index: 0机构: Ist Sci San Raffaele, Milan, Italy Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandOdore, Elodie论文数: 0 引用数: 0 h-index: 0机构: Hop Rene Huguenin, Inst Curie, St Cloud, France Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandRezai, Keyvan论文数: 0 引用数: 0 h-index: 0机构: Hop Rene Huguenin, Inst Curie, St Cloud, France Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandBernasconi, Elena论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandCascione, Luciano论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland Oncol Inst Southern Switzerland IOSI, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandRinaldi, Andrea论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandStathis, Anastasios论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst Southern Switzerland IOSI, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandRiveiro, Eugenia论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandCvitkovic, Esteban论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandZucca, Emanuele论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst Southern Switzerland IOSI, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, SwitzerlandBertoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland Oncol Inst Southern Switzerland IOSI, Bellinzona, Switzerland Inst Oncol Res IOR, Lymphoma & Genom Res Program, Bellinzona, Switzerland
- [2] OTX015 (MK-8628), a novel BET inhibitor, displays in vitro and in vivo antitumor effects alone and in combination with conventional therapies in glioblastoma models[J]. INTERNATIONAL JOURNAL OF CANCER, 2016, 139 (09) : 2047 - 2055Berenguer-Daize, Caroline论文数: 0 引用数: 0 h-index: 0机构: Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceAstorgues-Xerri, Lucile论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceOdore, Elodie论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Rene Huguenin Hosp, Inst Curie, Dept Radio Pharmacol, 35 Rue Daily, F-92210 St Cloud, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceCayol, Mylene论文数: 0 引用数: 0 h-index: 0机构: Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceCvitkovic, Esteban论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Oncoethix GmbH, Weystr 20, CH-6000 Luzern, Switzerland Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceNoel, Kay论文数: 0 引用数: 0 h-index: 0机构: Oncoethix GmbH, Weystr 20, CH-6000 Luzern, Switzerland Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceBekradda, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceMacKenzie, Sarah论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceRezai, Keyvan论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Inst Curie, Dept Radio Pharmacol, 35 Rue Daily, F-92210 St Cloud, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceLokiec, Francois论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Inst Curie, Dept Radio Pharmacol, 35 Rue Daily, F-92210 St Cloud, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceRiveiro, Maria E.论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, FranceOuafik, L'Houcine论文数: 0 引用数: 0 h-index: 0机构: Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, France Aix Marseille Univ, INSERM, CRO2, UMR S 911, F-13385 Marseille, France
- [3] Promising in vivo efficacy of the BET bromodomain inhibitor OTX015/MK-8628 in malignant pleural mesothelioma xenografts[J]. INTERNATIONAL JOURNAL OF CANCER, 2017, 140 (01) : 197 - 207Vazquez, Ramiro论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyLicandro, Simonetta Andrea论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyAstorgues-Xerri, Lucile论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyLettera, Emanuele论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyPanini, Nicolo论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyRomano, Michela论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyErba, Eugenio论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyUbezio, Paolo论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyBello, Ezia论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyLibener, Roberta论文数: 0 引用数: 0 h-index: 0机构: SS Antonio & Biagio & Cesare Arrigo Gen Hosp, Pathol Unit, Cytogenet & Mol Pathol Lab, Oncol, Alessandria, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyOrecchia, Sara论文数: 0 引用数: 0 h-index: 0机构: SS Antonio & Biagio & Cesare Arrigo Gen Hosp, Pathol Unit, Cytogenet & Mol Pathol Lab, Oncol, Alessandria, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyGrosso, Federica论文数: 0 引用数: 0 h-index: 0机构: SS Antonio & Biagio & Cesare Arrigo Gen Hosp, Pathol Unit, Cytogenet & Mol Pathol Lab, Oncol, Alessandria, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyRiveiro, Maria Eugenia论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyCvitkovic, Esteban论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Oncoethix GmbH, Luzern, Switzerland IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyBekradda, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyD'Incalci, Maurizio论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, ItalyFrapolli, Roberta论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy IRCCS Ist Ric Farmacol Mario Negri, Lab Canc Pharmacol, Via Giuseppe La Masa 19, I-20156 Milan, Italy
- [4] The BRD-inhibitor OTX015 Shows Pre-clinical Activity in Diffuse Large B-cell Lymphoma (DLBCL)[J]. EUROPEAN JOURNAL OF CANCER, 2012, 48 : 163 - 163Bonetti, P.论文数: 0 引用数: 0 h-index: 0机构: Oncol Res Inst, Bellinzona, Switzerland Oncol Res Inst, Bellinzona, SwitzerlandPonzoni, M.论文数: 0 引用数: 0 h-index: 0机构: Ist Sci San Raffaele, Milan, Italy Oncol Res Inst, Bellinzona, SwitzerlandTibiletti, M. G.论文数: 0 引用数: 0 h-index: 0机构: Insubria Univ, Varese, Italy Oncol Res Inst, Bellinzona, SwitzerlandStathis, A.论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst So Switzerland, Bellinzona, Switzerland Oncol Res Inst, Bellinzona, SwitzerlandHeirat, P.论文数: 0 引用数: 0 h-index: 0机构: Onocethix SA, Lausanne, SA, Switzerland Oncol Res Inst, Bellinzona, SwitzerlandZucca, E.论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst So Switzerland, Bellinzona, Switzerland Oncol Res Inst, Bellinzona, SwitzerlandBertoni, F.论文数: 0 引用数: 0 h-index: 0机构: Oncol Res Inst, Bellinzona, Switzerland Oncol Res Inst, Bellinzona, Switzerland
- [5] Activity of OTX015 (MK-8628), a BET-Bromodomain Inhibitor, in Acute Myeloid Leukemia (AML) Progenitor Cells[J]. BLOOD, 2015, 126 (23)Roulin, Louise论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceAli, Ashfaq论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceMasse, Aline论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceCoude, Marie-Magdelaine论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceBluteau, Dominique论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceBraun, Thorsten论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France CHU Avicenne, Clin Hematol, Bobigny, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceBerrou, Jeanning论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceBluteau, Olivier论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceDelord, Marc论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Bioinformat, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceRiveiro, Maria Eugenia论文数: 0 引用数: 0 h-index: 0机构: OTD, Clichy, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceHerait, Patrice Edouard论文数: 0 引用数: 0 h-index: 0机构: ONCOETHIX, Soisy Sous Montmorency, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceSoulier, Jean论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Diderot, Inst Hematol, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceBaruchel, Andre论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France Hop Robert Debre, Dept Hematol, F-75019 Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceGardin, Claude论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France Univ Paris 13, Avicenne Hosp, AP HP, Dept Hematol, Bobigny, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceDombret, Herve论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, Inst Univ Hematol, Lab Transfert Leucemies, Paris, France Hop St Louis, Dept Hematol, Leukemia Unit, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, FranceItzykson, Raphael论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, France Univ Paris 07, St Louis Hosp, Dept Hematol, Paris, France Univ Paris 07, St Louis Inst, INSERM, UMR7212 U944, Paris, France
- [6] Insights into the cellular pharmacological properties of the BET-inhibitor OTX015/MK-8628 (birabresib), alone and in combination, in leukemia models[J]. LEUKEMIA & LYMPHOMA, 2019, 60 (12) : 3067 - 3070Astorgues-Xerri, Lucile论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceVazquez, Ramiro论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, Bellinzona, Switzerland Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceOdore, Elodie论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Curie Inst, RadioPharmacol Dept, St Cloud, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceRezai, Keyvan论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Curie Inst, RadioPharmacol Dept, St Cloud, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceKahatt, Carmen论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceMackenzie, Sarah论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceBekradda, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceCoude, Marie-Magdelaine论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Diderot, Lab Transfert Leucemies, Paris, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceDombret, Herve论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Diderot, Lab Transfert Leucemies, Paris, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceGardin, Claude论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Diderot, Lab Transfert Leucemies, Paris, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceLokiec, Francois论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Curie Inst, RadioPharmacol Dept, St Cloud, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceRaymond, Eric论文数: 0 引用数: 0 h-index: 0机构: CHU Vaudois, Med Oncol Dept, Lausanne, Switzerland Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceNoel, Kay论文数: 0 引用数: 0 h-index: 0机构: Oncoethix SA, Luzern, Switzerland Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceCvitkovic, Esteban论文数: 0 引用数: 0 h-index: 0机构: Oncoethix SA, Luzern, Switzerland Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceHerait, Patrice论文数: 0 引用数: 0 h-index: 0机构: Oncoethix SA, Luzern, Switzerland Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceBertoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: Univ Svizzera Italiana, Inst Oncol Res, Bellinzona, Switzerland Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, FranceRiveiro, Maria E.论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France Oncol Therapeut Dev, 100 Rue Martre, F-92110 Clichy, France
- [7] BET Bromodomain Inhibitor OTX015 Affects the Expression of Micrornas Involved in the Pathogenesis of Diffuse Large B-Cell Lymphoma[J]. BLOOD, 2014, 124 (21)Cascione, Luciano论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOSI Oncol Inst Southern Switzerland, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandGaudio, Eugenio论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandBernasconi, Elena论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandTarantelli, Chiara论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandRinaldi, Andrea论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandTestoni, Monica论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandBomben, Riccardo论文数: 0 引用数: 0 h-index: 0机构: IRCCS, Ctr Riferimento Oncol, Aviano, PN, Italy IOR, Bellinzona, SwitzerlandGattei, Valter论文数: 0 引用数: 0 h-index: 0机构: Ctr Riferimento Oncol, I-33081 Aviano, Italy IOR, Bellinzona, SwitzerlandKwee, Ivo论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland Dalle Molle Inst Artificial Intelligence, Manno, Switzerland IOR, Bellinzona, SwitzerlandStathis, Anastasios论文数: 0 引用数: 0 h-index: 0机构: IOSI Oncol Inst Southern Switzerland, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandRiveiro, Maria Eugenia论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France IOR, Bellinzona, SwitzerlandZucca, Emanuele论文数: 0 引用数: 0 h-index: 0机构: IOSI Oncol Inst Southern Switzerland, Bellinzona, Switzerland IOR, Bellinzona, SwitzerlandBertoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: IOR, Bellinzona, Switzerland IOSI Oncol Inst Southern Switzerland, Bellinzona, Switzerland IOR, Bellinzona, Switzerland
- [8] OTX015 (MK-8628), a novel BET inhibitor, exhibits antitumor activity in non-small cell and small cell lung cancer models harboring different oncogenic mutations[J]. ONCOTARGET, 2016, 7 (51) : 84675 - 84687Riveiro, Maria E.论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Oncol Therapeut Dev, Clichy, FranceAstorgues-Xerri, Lucile论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Oncol Therapeut Dev, Clichy, FranceVazquez, Ramiro论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Milan, Italy Oncol Therapeut Dev, Clichy, FranceFrapolli, Roberta论文数: 0 引用数: 0 h-index: 0机构: IRCCS Ist Ric Farmacol Mario Negri, Milan, Italy Oncol Therapeut Dev, Clichy, FranceKwee, Ivo论文数: 0 引用数: 0 h-index: 0机构: IOR Inst Oncol Res, Lymphoma & Genom Res Program, Bellinzona, Switzerland SIB, Lausanne, Switzerland Oncol Therapeut Dev, Clichy, FranceRinaldi, Andrea论文数: 0 引用数: 0 h-index: 0机构: IOR Inst Oncol Res, Lymphoma & Genom Res Program, Bellinzona, Switzerland Oncol Therapeut Dev, Clichy, FranceOdore, Elodie论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Inst Curie, Radiopharmacol Dept, St Cloud, France Oncol Therapeut Dev, Clichy, FranceRezai, Keyvan论文数: 0 引用数: 0 h-index: 0机构: Rene Huguenin Hosp, Inst Curie, Radiopharmacol Dept, St Cloud, France Oncol Therapeut Dev, Clichy, FranceBekradda, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Oncol Therapeut Dev, Clichy, FranceInghirami, Giorgio论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Dept Pathol & Lab Med, New York, NY USA NYU, Sch Med, Dept Pathol, New York, NY USA NYU, Sch Med, Ctr Canc, New York, NY USA Oncol Therapeut Dev, Clichy, FranceD'Incalci, Maurizio论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, FranceNoel, Kay论文数: 0 引用数: 0 h-index: 0机构: Oncoethix SA, Oncoethix GmbH, Luzern, Switzerland Oncol Therapeut Dev, Clichy, FranceCvitkovic, Esteban论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Oncoethix SA, Oncoethix GmbH, Luzern, Switzerland Oncol Therapeut Dev, Clichy, FranceRaymond, Eric论文数: 0 引用数: 0 h-index: 0机构: CHU Vaudois, Dept Med Oncol, Lausanne, Switzerland Oncol Therapeut Dev, Clichy, FranceBertoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: IOR Inst Oncol Res, Lymphoma & Genom Res Program, Bellinzona, Switzerland Oncol Inst Southern Switzerland IOSI, Bellinzona, Switzerland Oncol Therapeut Dev, Clichy, France
- [9] Therapeutic efficacy of the bromodomain inhibitor OTX015/MK-8628 in ALK-positive anaplastic large cell lymphoma: an alternative modality to overcome resistant phenotypes[J]. ONCOTARGET, 2016, 7 (48) : 79623 - 79639Boi, Michela论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, Italy Univ Torino, Ctr Expt Res & Med Studies CeRMS, Turin, Italy Weill Cornell Med Coll, Dept Pathol & Lab Med, New York, NY 10065 USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyTodaro, Maria论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, Italy Univ Torino, Ctr Expt Res & Med Studies CeRMS, Turin, Italy Weill Cornell Med Coll, Dept Pathol & Lab Med, New York, NY 10065 USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyVurchio, Valentina论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, Italy Univ Torino, Ctr Expt Res & Med Studies CeRMS, Turin, Italy Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyYang, Shao Ning论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Joan & Sanford I Weill Dept Med, New York, NY USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyMoon, John论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Joan & Sanford I Weill Dept Med, New York, NY USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyKwee, Ivo论文数: 0 引用数: 0 h-index: 0机构: IOR Inst Oncol Res, Lymphoma & Genom Res Program, Bellinzona, Switzerland Dalle Molle Inst Artificial Intelligence IDSIA, Manno, Switzerland SIB, Lausanne, Switzerland Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyRinaldi, Andrea论文数: 0 引用数: 0 h-index: 0机构: IOR Inst Oncol Res, Lymphoma & Genom Res Program, Bellinzona, Switzerland Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyPan, Heng论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Dept Physiol & Biophys, Inst Computat Biomed, New York, NY USA Weill Cornell Med Coll, Inst Precis Med, New York, NY USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyCrescenzo, Ramona论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, Italy Univ Torino, Ctr Expt Res & Med Studies CeRMS, Turin, Italy Weill Cornell Med Coll, Dept Pathol & Lab Med, New York, NY 10065 USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyCheng, Mangeng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Lab, Vitro Pharmacol, Boston, MA USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyCerchietti, Leandro论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Joan & Sanford I Weill Dept Med, New York, NY USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyElemento, Olivier论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, Dept Physiol & Biophys, Inst Computat Biomed, New York, NY USA Weill Cornell Med Coll, Inst Precis Med, New York, NY USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyRiveiro, Maria E.论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyCvitkovic, Esteban论文数: 0 引用数: 0 h-index: 0机构: Oncol Therapeut Dev, Clichy, France Oncoethix SA, Luzern, Switzerland Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyBertoni, Francesco论文数: 0 引用数: 0 h-index: 0机构: IOR Inst Oncol Res, Lymphoma & Genom Res Program, Bellinzona, Switzerland IOSI Oncol Inst So Switzerland, Bellinzona, Switzerland Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, ItalyInghirami, Giorgio论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, Italy Univ Torino, Ctr Expt Res & Med Studies CeRMS, Turin, Italy Weill Cornell Med Coll, Dept Pathol & Lab Med, New York, NY 10065 USA NYU, Sch Med, Dept Pathol, New York, NY 10003 USA NYU, Sch Med, NYU Canc Ctr, New York, NY 10003 USA Univ Torino, Dept Mol Biotechnol & Hlth Sci, Turin, Italy
- [10] The BET Inhibitor OTX015 Exhibits In Vitro and In Vivo Antitumor Activity in Pediatric Ependymoma Stem Cell Models[J]. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 22 (04) : 1 - 19Servidei, Tiziana论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyMeco, Daniela论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyMartini, Maurizio论文数: 0 引用数: 0 h-index: 0机构: Univ Cattolica Sacro Cuore, Dept Pathol, Fdn Policlin Univ A Gemelli IRCCS, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyBattaglia, Alessandra论文数: 0 引用数: 0 h-index: 0机构: Univ Cattolica Sacro Cuore, Sect Gynecol & Obstet, Dept Life Sci & Publ Hlth, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyGranitto, Alessia论文数: 0 引用数: 0 h-index: 0机构: Univ Cattolica Sacro Cuore, Dept Pathol, Fdn Policlin Univ A Gemelli IRCCS, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyBuzzonetti, Alexia论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Oncol Gynecol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyBabini, Gabriele论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Oncol Gynecol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyMassimi, Luca论文数: 0 引用数: 0 h-index: 0机构: Univ Cattolica Sacro Cuore, Fdn Policlin Univ A Gemelli IRCCS, UOC Neurochirurg Infantile, Dipartimento Sci Invecchiamento Neurol Ortoped &, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyTamburrini, Gianpiero论文数: 0 引用数: 0 h-index: 0机构: Univ Cattolica Sacro Cuore, Fdn Policlin Univ A Gemelli IRCCS, UOC Neurochirurg Infantile, Dipartimento Sci Invecchiamento Neurol Ortoped &, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyScambia, Giovanni论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Oncol Gynecol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyRuggiero, Antonio论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, ItalyRiccardi, Riccardo论文数: 0 引用数: 0 h-index: 0机构: Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, Italy Fdn Policlin Univ A Gemelli IRCCS, Dept Woman & Child Hlth & Publ Hlth, UOC Pediat Oncol, I-00168 Rome, Italy