共 11 条
- [1] A novel class of selective estrogen receptors degraders regresses tumors in pre-clinical models of endocrine-resistant breast cancerCANCER RESEARCH, 2014, 74 (19)Joseph, James D.Darimont, BeatriceGovek, StevenBrigham, DanQian, JingSensintaffar, JohnShao, GangAparicio, AnnaKahraman, MehmetLai, AndiliyLee, Kyoung-JinLu, NhinNagasawa, JohnnyMoon, MichaelRix, PeterSmith, NickHager, Jeff
- [2] A novel class of selective estrogen receptors degraders regresses tumors in pre-clinical models of endocrine-resistant breast cancerCLINICAL CANCER RESEARCH, 2012, 18 (10)Darimont, BeatriceGovek, StevenLu, NihnNagasawa, JohnnyPrudente, ReneQian, JingSensintaffar, JohnShao, GangHeyman, RichardRix, PeterSmith, NicholasHager, JeffreyJoseph, JamesGrillot, KatherineAparicio, AnnaBischoff, EricKahraman, MehmetKaufman, JoshLai, AndiliyLee, Kyoung-Jin
- [3] Novel selective estrogen receptors degraders regress tumors in pre-clinical models of endocrine-resistant breast cancerCANCER RESEARCH, 2012, 72Hager, J. H.Darimont, B.Joseph, J.Govek, S.Grillot, K.Aparicio, A.Bischoff, E.Kahraman, M.Kaufman, J.Lai, A.Lee, K-JLu, N.Nagasawa, J.Prudente, R.Qian, J.Sensintaffar, J.Shao, G.Heyman, R.Rix, P.Smith, N. D.
- [4] A novel class of selective estrogen receptor degraders display activity in pre-clinical models of ERα plus ovarian cancerCLINICAL CANCER RESEARCH, 2013, 19Joseph, James D.Darimont, BeatriceGovek, StevenBrigham, DanAparicio, AnnaKahraman, MehmetLai, AndiliyLu, Lee NhinNagasawa, JohnnyKaufman, JoshMoon, MichaelPrudente, ReneQian, JingSensintaffar, JohnShao, GangRix, PeterSmith, NickHager, Jeff
- [5] Discovery of novel covalent selective estrogen receptor degraders against endocrine-resistant breast cancerActa Pharmaceutica Sinica B, 2023, (12) : 4963 - 4982Yubo WangJian MinXiangping DengTian FengHebing HuXinyi GuoYan ChengBaohua XieYu YangChun-Chi ChenRey-Ting GuoChune DongHai-Bing Zhou
- [6] Discovery of novel covalent selective estrogen receptor degraders against endocrine-resistant breast cancerACTA PHARMACEUTICA SINICA B, 2023, 13 (12) : 4963 - 4982Wang, YuboMin, JianDeng, XiangpingFeng, TianHu, HebingGuo, XinyiCheng, YanXie, BaohuaYang, YuChen, Chun-ChiGuo, Rey-TingDong, ChuneZhou, Hai-Bing
- [7] Discovery of a Novel Class of PROTACs as Potent and Selective Estrogen Receptor α Degraders to Overcome Endocrine-Resistant Breast Cancer In Vitro and In VivoJOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (10) : 6631 - 6651Xie, BaohuaYin, ZhinangHu, ZhiyeLv, JunhuiDu, ChuanqianDeng, XiangpingHuang, YuanLi, QiuziHuang, JianLiang, KaiweiZhou, Hai-BingDong, Chune
- [8] Discovery of Novel ERα and Aromatase Dual-Targeting PROTAC Degraders to Overcome Endocrine-Resistant Breast CancerJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (11) : 8913 - 8931Xin, LilanWang, ChaoCheng, YanWang, HongliGuo, XinyiDeng, XiaofeiDeng, XiangpingXie, BaohuaHu, HankunMin, ChangDong, ChuneZhou, Hai-Bing
- [9] Discovery of Thiochroman Derivatives as Potent, Oral Selective Estrogen Receptor Degraders and Antagonists for the Treatment of Endocrine-Resistant Breast CancerJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (23) : 21545 - 21567Zhang, DanLu, ZhengyuHe, YongqiLeng, Xin-YuMeng, XinLei, XiangKong, DeyuSun, LuluHu, WenhaoYang, Yushe
- [10] Discovery of GDC-0810 a novel, non-steroidal selective estrogen receptor degrader with robust activity in pre-clinical models of endocrine-resistant breast cancerCANCER RESEARCH, 2015, 75Joseph, JamesGovek, StevenDarimont, BeatriceBrigham, DanielAparicio, AnnaBischoff, EricKahraman, MehmetNannini, MichelleKaufman, JoshuaLai, AndilyLee, Kyoung-JinOeh, JasonLu, NhinZhou, WeiMoon, MichaelQian, JingSensintaffar, JohnShao, GangSampath, DeepakFriedman, Lori S.Rix, PeterHeyman, Richard A.Smith, NicholasHager, Jeffrey H.