Labeling of the high-affinity vasopressin subtype 1a receptor ligand, AVN778, with carbon-11 and evaluation as a candidate PET radioligand in monkey

被引:0
|
作者
Telu, Sanjay [1 ]
Xu Rong [1 ]
Liow, Jeih-San [1 ]
Gladding, Robert L. [1 ]
Zoghbi, Sami S. [1 ]
Guillon, Christophe D. [2 ,3 ]
Fabio, Karine M. [3 ]
Lu Shifang [2 ,4 ]
Heindel, Ned [3 ]
Simon, Neal [2 ,4 ]
Brownstein, Michael J. [2 ]
Innis, Robert B. [1 ]
Pike, Victor W. [1 ]
机构
[1] NIMH, Mol Imaging Branch, NIH, Bethesda, MD 20892 USA
[2] Azevan Pharmaceut Inc, Bethlehem, PA USA
[3] Lehigh Univ, Dept Chem, Bethlehem, PA 18015 USA
[4] Lehigh Univ, Dept Biol Sci, Bethlehem, PA 18015 USA
关键词
ANTAGONISTS;
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
P240
引用
收藏
页码:S327 / S327
页数:1
相关论文
共 11 条
  • [1] Labeling of FPEB with carbon-11 for evaluation as an mGluR5 radioligand in monkey with PET
    Simeon, Fabrice G.
    Yi Zhang
    Morse, Cheryl L.
    Yoo, Chul H.
    Gladding, Robert L.
    Fujita, Masahiro
    Innis, Robert B.
    Pike, Victor W.
    [J]. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2013, 56 : S329 - S329
  • [2] LABELING OF SP203 WITH CARBON-11 FOR EVALUATION AS AN MGLUR5 RADIOLIGAND IN MONKEY WITH PET
    Simeon, F. G.
    Hong, J.
    Liow, J.
    Gladding, R.
    Innis, R. B.
    Pike, V. W.
    [J]. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2009, 52 : S387 - S387
  • [3] Labeling of a new high-affinity TSPO PET radioligand in a pendant aryl trifluoromethyl group with either carbon-11 or fluorine-18
    Simeon, Fabrice
    Yang, Bo Yeun
    Telu, Sanjay
    Taliani, Sabrina
    Castellano, Sabrina
    Da Settimo, Federico
    Pike, Victor
    [J]. JOURNAL OF NUCLEAR MEDICINE, 2017, 58
  • [4] Synthesis and evaluation of a carbon-11 labeled PET-radioligand with affinity for the transient receptor potential vanilloid subfamily type 1 receptor.
    Van Veghel, D.
    Cleynhens, J.
    Van Laere, K.
    Voets, T.
    Verbruggen, A.
    Bormans, G.
    [J]. EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2009, 36 (SUPPL 2) : 236 - 237
  • [5] Synthesis and evaluation of a carbon-11 labeled PET-radioligand with affinity for the transient receptor potential vanilloid subfamily type 1 receptor.
    Van Veghel, D.
    Cleynhens, J.
    Van Laere, K.
    Voets, T.
    Verbruggen, A.
    Bormans, G.
    [J]. EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2009, 36 : S236 - S237
  • [6] CARBON-11 LABELING AND PRELIMINARY EVALUATION OF SSR180575, A HIGHLY PROMISING RADIOLIGAND FOR IMAGING THE PERIPHERAL BENZODIAZEPINE RECEPTOR WITH PET
    Dolle, F.
    Boutin, H.
    Thominiaux, C.
    Chauveau, F.
    Boisgard, R.
    Demphel, S.
    Roy, S.
    Boisnard, S.
    Rooney, T.
    Benavides, J.
    Hantraye, P.
    Tavitian, B.
    [J]. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2009, 52 : S93 - S93
  • [7] Two new C-methyl analogues of WAY-100635-preparation, labeling with carbon-11 and evaluation as PET radioligands for brain 5-HT1A receptors in monkey
    Pike, VW
    Tarkiainen, J
    Marchais, S
    McCarron, JA
    Halldin, C
    Sovago, J
    Gulyas, B
    Truong, P
    Wikstrom, HV
    Farde, L
    [J]. NEUROIMAGE, 2002, 16 (03) : S19 - S19
  • [8] Radiosynthesis and Evaluation of [11C]3-Hydroxycyclopent-1-enecarboxylic Acid as Potential PET Ligand for the High-Affinity γ-Hydroxybutyric Acid Binding Sites
    Jensen, Claus H.
    Hansen, Hanne D.
    Bay, Tina
    Vogensen, Stine B.
    Lehel, Szabolcs
    Thiesen, Louise
    Bundgaard, Christoffer
    Clausen, Rasmus P.
    Knudsen, Gitte M.
    Herth, Matthias M.
    Wellendorph, Petrine
    Frolund, Bente
    [J]. ACS CHEMICAL NEUROSCIENCE, 2017, 8 (01): : 22 - 27
  • [9] Radiosynthesis and Evaluation in Monkey of Three C-11-Labeled 1,5-Diarylpyrazoles as High Potency Candidate PET Radioligands for Cannabinoid Subtype-1 Receptors in Brain
    Donohue, Sean R.
    Zoghbi, Sami S.
    Yasuno, Fumihiko
    Terry, Garth
    Gourley, Jonathan P.
    Innis, Robert B.
    Halldin, Christer
    Pike, Victor W.
    [J]. CURRENT RADIOPHARMACEUTICALS, 2008, 1 (02) : 93 - 102
  • [10] Quantification of PET studies with the very high-affinity dopamine D2/D3 receptor ligand [11C]FLB 457:: re-evaluation of the validity of using a cerebellar reference region
    Asselin, Marie-Claude
    Montgomery, Andrew J.
    Grasby, Paul M.
    Hume, Susan P.
    [J]. JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM, 2007, 27 (02): : 378 - 392