Development of a new cascade reaction for convergent synthesis of pyrazolo[1,5-a]quinoline derivatives under transition-metal-free conditions

被引：17
|
作者：
Kato, Jun-ya [1 ]
Aoyama, Hiroshi [1 ]
Yokomatsu, Tsutomu [1 ]
机构：
[1] Tokyo Univ Pharm & Life Sci, Sch Pharm, Hachioji, Tokyo 1920392, Japan
来源：
ORGANIC & BIOMOLECULAR CHEMISTRY | 2013年 / 11卷 / 07期
关键词：
CYCLOADDITION; RECEPTOR;
D O I：
10.1039/c2ob27050a
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A novel method for the synthesis of pyrazolo[1,5-a]quinolines under the transition-metal-free conditions has been developed. This method involves a novel combination of aromatic nucleophilic substitution and Knoevenagel condensation reactions to give pyrazolo[1,5-a]quinolines.
引用
收藏
页码：1171 / 1178
页数：8
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