Novel nonsedative agents to treat epilepsy: Benzodiazepine-related ligands that do not develop tolerance

被引:0
|
作者
Edwankar, Rahul V. [1 ]
Edwankar, Chitra R. [1 ]
Stables, James P. [2 ]
Roth, Bryan L. [3 ,4 ]
Furtmueller, Roman [5 ]
Sieghart, Werner [6 ]
Cook, James M. [1 ]
机构
[1] Univ Wisconsin, Dept Chem & Biochem, Milwaukee, WI 53211 USA
[2] NINDS, Epilepsy Branch, NIH, Rockville, MD 20852 USA
[3] Univ N Carolina, NIMH, Psychoact Drug Screening Program, Chapel Hill, NC 27599 USA
[4] Univ N Carolina, Dept Pharmacol, Chapel Hill, NC 27599 USA
[5] Med Univ Vienna, Ctr Brain Res, A-1090 Vienna, Austria
[6] Med Univ, Brain Res Inst, A-1090 Vienna, Austria
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
99-MEDI
引用
收藏
页数:1
相关论文
共 7 条
  • [1] New benzodiazepine-related agents to treat neuropathic pain
    Edwankar, Chitra R.
    Edwankar, Rahul V.
    Zeilhofer, Hanns
    Stables, James P.
    Roth, Bryan L.
    Furtmueller, Roman
    Sieghart, Werner
    Cook, James M.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238
  • [2] NOVEL LONG-ACTING BENZODIAZEPINE RECEPTOR LIGANDS WITH POTENTIAL VALUE FOR THE TREATMENT OF EPILEPSY
    MOREAU, JL
    BONETTI, EP
    HUNKELER, W
    JENCK, F
    MARTIN, JR
    HAEFELY, WE
    PSYCHOPHARMACOLOGY, 1990, 101 : S39 - S39
  • [3] Several New Diverse Anticonvulsant Agents Discovered in a Virtual Screening Campaign Aimed at Novel Antiepileptic Drugs to Treat Refractory Epilepsy
    Di Ianni, Mauricio E.
    Enrique, Andrea V.
    Palestro, Pablo H.
    Gavernet, Luciana
    Talevi, Alan
    Bruno-Blanch, Luis E.
    JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2012, 52 (12) : 3325 - 3330
  • [4] Improved Synthesis of Anxiolytic, Anticonvulsant, and Antinociceptive α2/α3-GABA(A)-ergic Receptor Subtype Selective Ligands as Promising Agents to Treat Anxiety, Epilepsy, and Neuropathic
    Li, Guanguan
    Golani, Lalit K.
    Jahan, Rajwana
    Rashid, Farjana
    Cook, James M.
    SYNTHESIS-STUTTGART, 2018, 50 (20): : 4124 - 4132
  • [5] SYNTHESIS AND PRELIMINARY EVALUATION OF PYRAZOLO[1,5-A]PYRIDO[3,4-E]PYRIMIDIN-6(7H)-ONES AND RELATED-COMPOUNDS, AS BENZODIAZEPINE RECEPTOR LIGANDS AND ANTICONVULSANT AGENTS
    SELLERI, S
    BRUNI, F
    COSTANZO, A
    GUERRINI, G
    AIELLO, PM
    IAVARONE, G
    MARTINI, C
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 1992, 27 (09) : 985 - 990
  • [6] Long-term studies on anticonvulsant tolerance and withdrawal characteristics of benzodiazepine receptor ligands in different seizure models in mice .2. The novel imidazoquinazolines NNC 14-0185 and NNC 14-0189
    Loscher, W
    Rundfeldt, C
    Honack, D
    Ebert, U
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1996, 279 (02): : 573 - 581
  • [7] MOLECULAR RECOGNITION BETWEEN LIGANDS AND NUCLEIC-ACIDS - NOVEL PYRIDINE-CONTAINING AND BENZOXAZOLE-CONTAINING AGENTS RELATED TO HOECHST-33258 THAT EXHIBIT ALTERED DNA-SEQUENCE SPECIFICITY DEDUCED FROM FOOTPRINTING ANALYSIS AND SPECTROSCOPIC STUDIES
    BATHINI, Y
    RAO, KE
    SHEA, RG
    LOWN, JW
    CHEMICAL RESEARCH IN TOXICOLOGY, 1990, 3 (03) : 268 - 280