A NEW SYNTHESIS OF AMINO SUBSTITUTED AZOLO[1,3,5]TRIAZINES VIA REACTION OF N1,N1-DIMETHYL-N2-AZOLYLFORMAMIDINES WITH CYANAMIDE

被引：23

作者：

Kalinin, Dmitrii V. ^{[1
]}

Kalinina, Svetlana A. ^{[1
]}

Dolzhenko, Anton V. ^{[2
,3
]}

机构：

[1] Perm State Pharmaceut Acad, Perm 614990, Russia

[2] Monash Univ, Jeffrey Cheah Sch Med & Hlth Sci, Bandar Sunway 46150, Selangor, Malaysia

[3] Curtin Univ Technol, Sch Pharm, Curtin Hlth Innovat Res Inst, Perth, WA 6845, Australia

来源：

HETEROCYCLES | 2013年 / 87卷 / 01期

关键词：

Triazole; Pyrazole; Triazine; Formamidine; Benzimidazole; TAUTOMERISM; CHEMISTRY; ADENINE; ROUTE;

D O I：

10.3987/COM-12-12601

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The amino substituted triazine ring was annelated to aminoazoles using a new effective synthetic procedure. The method of preparation involved initial formation of azolylformamidines in the reaction of aminoazoles with N,N-dimethylformamide dimethyl acetal followed by the triazine ring closure with cyanamide affording therefore fused aminotriazines.

引用

页码：147 / 154

页数：8

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