Synthesis of pyrido[1,2-a]benzimidazoles and other fused imidazole derivatives with a bridgehead nitrogen atom

被引：15
|
作者：
Begunov, R. S. [1 ]
Ryzvanovich, G. A. [1 ]
机构：
[1] PG Demidov Yaroslavl State Univ, Ul Sovetskaya 14, Yaroslavl 150000, Russia
来源：
RUSSIAN CHEMICAL REVIEWS | 2013年 / 82卷 / 01期
关键词：
CONDENSED RING-SYSTEMS; POTENTIAL ANXIOLYTIC AGENTS; ONE-POT SYNTHESIS; HETEROATOMIC PHOTOCYCLIZATION; REGIOSELECTIVE SYNTHESIS; HETEROCYCLIC SYNTHESIS; ANTITUMOR-ACTIVITY; FACILE SYNTHESIS; ROUTE; 2-AMINOBENZIMIDAZOLE;
D O I：
10.1070/RC2013v082n01ABEH004295
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Main methods for the synthesis of fused imidazole derivatives with a bridgehead nitrogen atom are systematically considered and summarized. The reaction mechanisms that underlie the methods for the synthesis of pyrido[1,2-a]benzimidazoles and related compounds are described. Biological properties and mechanisms of the biological activity of fused azaheterocycles are discussed. The bibliography includes 152 references.
引用
收藏
页码：77 / 97
页数：21
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