Iminophosphoranes in heterocyclic chemistry. A simple one-pot synthesis of dihydropyrimidines and pyrimidines

被引:0
|
作者
Rossi, E [1 ]
Abbiati, G [1 ]
Pini, E [1 ]
机构
[1] Univ Milan, Fac Farm, Ist Chim Organ, I-20133 Milan, Italy
关键词
amidines; nitrogen-ylids; condensation reactions; dihydropyrimidines; 8pyrimidines;
D O I
暂无
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The condensation of N-triphenylphosphoraniliden-benzamidine with acyclic alpha,beta-unsaturated aldehydes produces dihydropyrimidines in good to high yields. The methodology has been extended to alicyclic and heterocyclic aldehydes.
引用
收藏
页码:1265 / 1267
页数:3
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