Three-Component Synthesis of Diaryl Propargylamines Catalyzed by Copper

被引：0

作者：

Liang, Linfeng ^{[1
]}

Liu, Jun ^{[1
]}

Xu, Xiaobing ^{[1
]}

Li, Yanzhong ^{[1
]}

机构：

[1] E China Normal Univ, Dept Chem, Shanghai 200062, Peoples R China

来源：

CHINESE JOURNAL OF ORGANIC CHEMISTRY | 2009年 / 29卷 / 10期

关键词：

three-component reaction; propargylamine; diarylamine; copper catalysis; C-H ACTIVATION; ALDEHYDE-ALKYNE-AMINE; EFFICIENT; CONDENSATION;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of new diaryl propargylamines were synthesized by the reaction of aldehyde, phenylacetylene and diarylamine, and structurally characterized by H-1 NMR, C-13 NMR and HRMS data.

引用

页码：1672 / 1675

页数：4

共 20 条

[1] Dyker G, 1999, ANGEW CHEM INT EDIT, V38, P1699, DOI 10.1002/(SICI)1521-3773(19990614)38:12<1698::AID-ANIE1698>3.0.CO
[2] 2-6
[3] Direct addition of TMS-acetylene to aldimines catalyzed by a simple, commercially available Ir(I) complex
Fischer, C
Carreira, EM
[J]. ORGANIC LETTERS, 2001, 3 (26) : 4319 - 4321
[4] Enantioselective, copper(I)-catalyzed three-component reaction for the preparation of propargylamines
Gommermann, N
Koradin, X
Polborn, K
Knochel, P
[J]. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2003, 42 (46) : 5763 - 5766
[5] Practical highly enantioselective synthesis of propargylamines through a copper-catalyzed one-pot three-component condensation reaction
Gommermann, Nina
Knochel, Paul
[J]. CHEMISTRY-A EUROPEAN JOURNAL, 2006, 12 (16) : 4380 - 4392
[6] Huma HZS, 2002, TETRAHEDRON LETT, V43, P6485
[7] STEREOSELECTIVE EPOXIDATION OF PHE-GLY AND PHE-PHE VINYL ISOSTERES
JENMALM, A
BERTS, W
LI, YL
LUTHMAN, K
CSOREGH, I
HACKSELL, U
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1994, 59 (05): : 1139 - 1148
[8] Kabalka GW, 2001, SYNLETT, P676
[9] Highly efficient Grignard-type imine additions via C-H activation in water and under solvent-free conditions
Li, CJ
Wei, CM
[J]. CHEMICAL COMMUNICATIONS, 2002, (03) : 268 - 269
[10] Li M, 2008, CHINESE J ORG CHEM, V28, P472

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