共 50 条
- [1] Engineering of highly potent and selective HNTX-III mutant against hNav1.7 sodium channel for treatment of painJOURNAL OF BIOLOGICAL CHEMISTRY, 2021, 296Zhang, Yunxiao论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Inst Sci & Technol, Sch Chem & Chem Engn, Key Lab Hunan Prov Adv Carbon Based Funct Mat, Yueyang, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaWang, Li论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaPeng, Dezheng论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Inst Sci & Technol, Sch Chem & Chem Engn, Key Lab Hunan Prov Adv Carbon Based Funct Mat, Yueyang, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaZhang, Qingfeng论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaYang, Qiuchu论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaLi, Jiayan论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaLi, Dan论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaTang, Dongfang论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaChen, Minzhi论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaLiang, Songping论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaLiu, Yu论文数: 0 引用数: 0 h-index: 0机构: Hunan Inst Sci & Technol, Sch Chem & Chem Engn, Key Lab Hunan Prov Adv Carbon Based Funct Mat, Yueyang, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaWang, Sheng论文数: 0 引用数: 0 h-index: 0机构: Huazhong Univ Sci & Technol, Coll Life Sci & Technol, Minist Educ, Key Lab Mol Biophys, Wuhan, Hubei, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R ChinaLiu, Zhonghua论文数: 0 引用数: 0 h-index: 0机构: Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China Hunan Normal Univ, Coll Life Sci, Natl & Local Joint Engn Lab Anim Peptide Drug Dev, Changsha, Hunan, Peoples R China
- [2] Engineering Highly Potent and Selective Microproteins against Nav1.7 Sodium Channel for Treatment of PainJOURNAL OF BIOLOGICAL CHEMISTRY, 2016, 291 (27) : 13974 - 13986Shcherbatko, Anatoly论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USARossi, Andrea论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAFoletti, Davide论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA 23andme, 899 W Evelyn Ave, Mountain View, CA 94041 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAZhu, Guoyun论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USABogin, Oren论文数: 0 引用数: 0 h-index: 0机构: Amunix, Mountain View, CA 94043 USA Chan Bio Ltd, IL-69416 Tel Aviv, Israel Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USACasas, Meritxell Galindo论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USARickert, Mathias论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Delinia Biosci, 953 Indiana St, San Francisco, CA USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAHasa-Moreno, Adela论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USABartsevich, Victor论文数: 0 引用数: 0 h-index: 0机构: Amunix, Mountain View, CA 94043 USA Precis BioSci, 302 E Pettigrew St, Durham, NC 27701 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USACrameri, Andreas论文数: 0 引用数: 0 h-index: 0机构: Amunix, Mountain View, CA 94043 USA GlaxoSmithKline, Stevenage SG1 2NY, Herts, England Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USASteiner, Alexander R.论文数: 0 引用数: 0 h-index: 0机构: Sutro Biopharma, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAHenningsen, Robert论文数: 0 引用数: 0 h-index: 0机构: Sutro Biopharma, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAGill, Avinash论文数: 0 引用数: 0 h-index: 0机构: Sutro Biopharma, San Francisco, CA 94080 USA Genentech Inc, 1DNA Way, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAPons, Jaume论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Alexo Therapeut, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAShelton, David L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USARajpal, Arvind论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Bristol Myers Squibb, 700 Bay Rd, Redwood City, CA 94063 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USAStrop, Pavel论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA Bristol Myers Squibb, 700 Bay Rd, Redwood City, CA 94063 USA Pfizer Inc, Rinat Labs, San Francisco, CA 94080 USA
- [3] Development of New Benzenesulfonamides As Potent and Selective Nav1.7 Inhibitors for the Treatment of PainJOURNAL OF MEDICINAL CHEMISTRY, 2017, 60 (06) : 2513 - 2525Wu, Yong-Jin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAGuernon, Jason论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAShi, Jianliang论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USADitta, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USARobbins, Kevin J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USARajamani, Ramkumar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAEaston, Amy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USANewton, Amy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USABourin, Clotilde论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAMosure, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USASoars, Matthew G.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAKnox, Ronald J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAMatchett, Michele论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAPieschl, Rick L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAPost-Munson, Debra J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAWang, Shuya论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAHerrington, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAGraef, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USANewberry, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USABristow, Linda J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAMeanwell, Nicholas A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAOlson, Richard论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USAThompson, Lorin A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USADzierba, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb Co, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA
- [4] Engineering Potent and Selective Analogues of GpTx-1, a Tarantula Venom Peptide Antagonist of the NaV1.7 Sodium ChannelJOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (05) : 2299 - 2314Murray, Justin K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USALigutti, Joseph论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USALiu, Dong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAZou, Anruo论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAPoppe, Leszek论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USALi, Hongyan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAAndrews, Kristin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAMoyer, Bryan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAMcDonough, Stefan I.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Neurosci, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAFavreau, Philippe论文数: 0 引用数: 0 h-index: 0机构: Atheris Labs, CH-1233 Geneva, Switzerland Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAStoecklin, Reto论文数: 0 引用数: 0 h-index: 0机构: Atheris Labs, CH-1233 Geneva, Switzerland Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USAMiranda, Les P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA
- [5] Evaluation of Selective NaV1.7 Inhibitors for the Treatment of Ocular PainINVESTIGATIVE OPHTHALMOLOGY & VISUAL SCIENCE, 2018, 59 (09)Delwig, Anton论文数: 0 引用数: 0 h-index: 0机构: SiteOne Therapeut, San Francisco, CA USA SiteOne Therapeut, San Francisco, CA USAPajouhesh, Hassan论文数: 0 引用数: 0 h-index: 0机构: SiteOne Therapeut, San Francisco, CA USA SiteOne Therapeut, San Francisco, CA USA论文数: 引用数: h-index:机构:Du Bois, Justin论文数: 0 引用数: 0 h-index: 0机构: SiteOne Therapeut, San Francisco, CA USA Stanford Univ, Palo Alto, CA 94304 USA SiteOne Therapeut, San Francisco, CA USAMiljanich, George论文数: 0 引用数: 0 h-index: 0机构: SiteOne Therapeut, San Francisco, CA USA SiteOne Therapeut, San Francisco, CA USAMulcahy, John论文数: 0 引用数: 0 h-index: 0机构: SiteOne Therapeut, San Francisco, CA USA SiteOne Therapeut, San Francisco, CA USA
- [6] Familial pain syndromes from mutations of the Nav1.7 sodium channelYEAR IN NEUROLOGY 2, 2010, 1184 : 196 - 207Fischer, Tanya Z.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Sch Med, Dept Neurol, New Haven, CT 06510 USA Yale Univ, Sch Med, Ctr Neurosci & Regenerat Res, New Haven, CT 06510 USA Vet Adm Connecticut Healthcare Syst, Rehabil Res Ctr, West Haven, CT USA Yale Univ, Sch Med, Dept Neurol, New Haven, CT 06510 USAWaxman, Stephen G.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Sch Med, Dept Neurol, New Haven, CT 06510 USA Yale Univ, Sch Med, Ctr Neurosci & Regenerat Res, New Haven, CT 06510 USA Vet Adm Connecticut Healthcare Syst, Rehabil Res Ctr, West Haven, CT USA Yale Univ, Sch Med, Dept Neurol, New Haven, CT 06510 USA
- [7] Discovery of PF-05089771: A potent, subtype selective Nav1.7 inhibitor for the treatment of painABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Swain, Nigel论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Worldwide Med Chem, Cambridge, England Pfizer, Worldwide Med Chem, Cambridge, England
- [8] Mechanism of inhibition by chlorpromazine of the human pain threshold sodium channel, Nav1.7NEUROSCIENCE LETTERS, 2017, 639 : 1 - 7Lee, Su-Jin论文数: 0 引用数: 0 h-index: 0机构: Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South Korea Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South KoreaKim, Dong-Hyun论文数: 0 引用数: 0 h-index: 0机构: Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South Korea Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South KoreaHahn, Sang June论文数: 0 引用数: 0 h-index: 0机构: Catholic Univ Korea, Coll Med, Dept Physiol, Seoul 06591, South Korea Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South KoreaWaxman, Stephen G.论文数: 0 引用数: 0 h-index: 0机构: Yale Univ, Sch Med, Dept Neurol, New Haven, CT 06510 USA Yale Univ, Sch Med, Ctr Neurosci & Regenerat Res, New Haven, CT 06510 USA VA Connecticut Healthcare Syst, Rehabil Res Ctr, West Haven, CT 06516 USA Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South KoreaChoi, Jin-Sung论文数: 0 引用数: 0 h-index: 0机构: Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South Korea Catholic Univ Korea, Coll Pharm, 43 Jibong Ro, Bucheon Si 14662, Gyeonggi Do, South Korea
- [9] Discovery of indole- and indazole-acylsulfonamides as potent and selective Nav1.7 inhibitors for the treatment of painABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256Luo, Guanglin论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAChen, Ling论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAEaston, Amy论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USANewton, Amy论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USABourin, Clotilde论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAShields, Eric论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAMosure, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USASoar, Mattew论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAKnox, Ronald论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAMatchett, Michele论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAPieschl, Rick论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAPost-Munson, Debra论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAWang, Shuya论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAHerrington, James论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAGraef, John论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USANewberry, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USABristow, Linda论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAMeanwell, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USAThompson, Lorin论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USADzierba, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Brisol Myers Squibb, Res & Dev, Princeton, NJ USA Brisol Myers Squibb, Res & Dev, Princeton, NJ USA
- [10] Discovery of Indole- and Indazole-acylsulfonamides as Potent and Selective NaV1.7 Inhibitors for the Treatment of PainJOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (02) : 831 - 856Luo, Guanglin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAChen, Ling论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAEaston, Amy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USANewton, Amy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USABourin, Clotilde论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAShields, Eric论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAMosure, Kathy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USASoars, Matthew G.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAKnox, Ronald J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAMatchett, Michele论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAPieschl, Rick L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAPost-Munson, Debra J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAWang, Shuya论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAHerrington, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAGraef, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USANewberry, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USASivarao, Digavalli V.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USASenapati, Arun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USABristow, Linda J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAMeanwell, Nicholas A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USAThompson, Lorin A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USADzierba, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, POB 4000, Princeton, NJ 08543 USA