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- [1] Discovery of a first-in-class reversible DNMT1-selective inhibitor with improved tolerability and efficacy in acute myeloid leukemiaNATURE CANCER, 2021, 2 (10) : 1002 - +Pappalardi, Melissa B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAKeenan, Kathryn论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USACockerill, Mark论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAKellner, Wendy A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAStowell, Alexandra论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USASherk, Christian论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAWong, Kristen论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAPathuri, Sarath论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Epigenet & Mol Carcinogenesis, Houston, TX 77030 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USABriand, Jacques论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USASteidel, Michael论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Funct Genom, Heidelberg, Germany GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAChapman, Philip论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAGroy, Arthur论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Future Pipeline Discovery, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAWiseman, Ashley K.论文数: 0 引用数: 0 h-index: 0机构: Van Andel Res Inst, Ctr Epigenet, Grand Rapids, MI USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMcHugh, Charles F.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USACampobasso, Nino论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAGraves, Alan P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAFairweather, Emma论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAWerner, Thilo论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Funct Genom, Heidelberg, Germany GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USARaoof, Ali论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAButlin, Roger J.论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USARueda, Lourdes论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAHorton, John R.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Epigenet & Mol Carcinogenesis, Houston, TX 77030 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAFosbenner, David T.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAZhang, Cunyu论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAHandler, Jessica L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMuliaditan, Morris论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Drug Metab & Pharmacokinet Modelling, Stevenage, Herts, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMebrahtu, Makda论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAJaworski, Jon-Paul论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMcNulty, Dean E.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USABurt, Charlotte论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAEberl, H. Christian论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Funct Genom, Heidelberg, Germany GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USATaylor, Amy N.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAHo, Thau论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMerrihew, Susan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAFoley, Shawn W.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USARutkowska, Anna论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Funct Genom, Heidelberg, Germany GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USALi, Mei论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USARomeril, Stuart P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAGoldberg, Kristin论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAZhang, Xing论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Epigenet & Mol Carcinogenesis, Houston, TX 77030 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAKershaw, Christopher S.论文数: 0 引用数: 0 h-index: 0机构: Univ Manchester, Drug Discovery Unit, Canc Res UK Manchester Inst, Alderley Pk, Macclesfield, Cheshire, England GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USABantscheff, Marcus论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Funct Genom, Heidelberg, Germany GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAJurewicz, Anthony J.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMinthorn, Elisabeth论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAGrandi, Paola论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Funct Genom, Heidelberg, Germany GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAPatel, Mehul论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Med Sci & Technol, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USABenowitz, Andrew B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Future Pipeline Discovery, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAMohammad, Helai P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAGilmartin, Aidan G.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Future Pipeline Discovery, Collegeville, PA USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USAPrinjha, Rab K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA GlaxoSmithKline, Canc Epigenet Res Unit, Oncol, Collegeville, PA 19426 USA
- [2] Discovery of a first-in-class reversible DNMT1-selective inhibitor with improved tolerability and efficacy in acute myeloid leukemiaNature Cancer, 2021, 2 : 1002 - 1017Melissa B. Pappalardi论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyKathryn Keenan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMark Cockerill论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyWendy A. Kellner论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAlexandra Stowell论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyChristian Sherk论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyKristen Wong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologySarath Pathuri论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyJacques Briand论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMichael Steidel论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyPhilip Chapman论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyArthur Groy论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAshley K. Wiseman论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyCharles F. McHugh论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyNino Campobasso论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAlan P. Graves论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyEmma Fairweather论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyThilo Werner论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAli Raoof论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyRoger J. Butlin论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyLourdes Rueda论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyJohn R. Horton论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyDavid T. Fosbenner论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyCunyu Zhang论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyJessica L. Handler论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMorris Muliaditan论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMakda Mebrahtu论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyJon-Paul Jaworski论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyDean E. McNulty论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyCharlotte Burt论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyH. Christian Eberl论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAmy N. Taylor论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyThau Ho论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologySusan Merrihew论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyShawn W. Foley论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAnna Rutkowska论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMei Li论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyStuart P. Romeril论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyKristin Goldberg论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyXing Zhang论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyChristopher S. Kershaw论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMarcus Bantscheff论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAnthony J. Jurewicz论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyElisabeth Minthorn论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyPaola Grandi论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyMehul Patel论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAndrew B. Benowitz论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyHelai P. Mohammad论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyAidan G. Gilmartin论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, OncologyRab K. Prinjha论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline,Cancer Epigenetics Research Unit, Oncology
- [3] Discovery of a first-in-class ERK 1,2 inhibitorMOLECULAR CANCER RESEARCH, 2014, 12Samatar, Ahmed A.论文数: 0 引用数: 0 h-index: 0
- [4] Discovery of the first-in-class SHP1 covalent inhibitor for cancer immunotherapyCANCER RESEARCH, 2024, 84 (06)Qu, Zihan论文数: 0 引用数: 0 h-index: 0Meke, Frederick Nguele论文数: 0 引用数: 0 h-index: 0Zhang, Zheng论文数: 0 引用数: 0 h-index: 0Bai, Yunpeng论文数: 0 引用数: 0 h-index: 0Krabill, Aaron D.论文数: 0 引用数: 0 h-index: 0Muli, Christine S.论文数: 0 引用数: 0 h-index: 0Jassim, Brenson A.论文数: 0 引用数: 0 h-index: 0Dong, Jiajun论文数: 0 引用数: 0 h-index: 0Li, Jinyue论文数: 0 引用数: 0 h-index: 0Yuyen, Nguyen论文数: 0 引用数: 0 h-index: 0Tao, Andy W.论文数: 0 引用数: 0 h-index: 0Trader, Darci T.论文数: 0 引用数: 0 h-index: 0Zhang, Zhong-Yin论文数: 0 引用数: 0 h-index: 0
- [5] Discovery of a first-in-class allosteric inhibitor of the small GTPase Rac1CANCER RESEARCH, 2024, 84 (06)Silverman, Robert论文数: 0 引用数: 0 h-index: 0Cooper, Alan论文数: 0 引用数: 0 h-index: 0Kar, Ronodip论文数: 0 引用数: 0 h-index: 0Raman, Mayuri V.论文数: 0 引用数: 0 h-index: 0Ravirala, Ramu论文数: 0 引用数: 0 h-index: 0Shah, Mubarak Hasan论文数: 0 引用数: 0 h-index: 0Mahankali, Sandeep论文数: 0 引用数: 0 h-index: 0Goka, Erik T.论文数: 0 引用数: 0 h-index: 0
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- [7] Discovery and Characterization of Selective, First-in-Class Inhibitors of Citron KinaseJOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (04) : 2631 - 2666Maw, Joshua J.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USACoker, Jesse A.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAArya, Tarun论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAGoins, Christopher M.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USASonawane, Dhiraj论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAHan, Sang Hoon论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USARees, Matthew G.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USARonan, Melissa M.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USARoth, Jennifer A.论文数: 0 引用数: 0 h-index: 0机构: Broad Inst MIT & Harvard, Cambridge, MA 02142 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAWang, Nancy S.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAHeemers, Hannelore V.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Dept Canc Biol, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAMacdonald, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USAStauffer, Shaun R.论文数: 0 引用数: 0 h-index: 0机构: Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA Cleveland Clin, Lerner Res Inst, Ctr Therapeut Discovery, Cleveland, OH 44195 USA
- [8] Discovery of a first-in-class EZH2 selective degraderNATURE CHEMICAL BIOLOGY, 2020, 16 (02) : 214 - +Ma, Anqi论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAStratikopoulos, Elias论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAPark, Kwang-Su论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAWei, Jieli论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAMartin, Tiphaine C.论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAYang, Xiaobao论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USASchwarz, Megan论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USALeshchenko, Violetta论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Med, Div Hematol & Oncol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USARialdi, Alexander论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USADale, Brandon论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USALagana, Alessandro论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Icahn Inst Data Sci & Genom Technol, Inst Next Generat Healthcare, Dept Genet & Genom Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAGuccione, Ernesto论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAParekh, Samir论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Med, Div Hematol & Oncol, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAParsons, Ramon论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USAJin, Jian论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Dept Pharmacol Sci, Mt Sinai Ctr Therapeut Discovery, New York, NY 10029 USA
- [9] Discovery of a first-in-class EZH2 selective degraderNature Chemical Biology, 2020, 16 : 214 - 222Anqi Ma论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesElias Stratikopoulos论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesKwang-Su Park论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesJieli Wei论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesTiphaine C. Martin论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesXiaobao Yang论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesMegan Schwarz论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesVioletta Leshchenko论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesAlexander Rialdi论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesBrandon Dale论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesAlessandro Lagana论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesErnesto Guccione论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesSamir Parekh论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesRamon Parsons论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological SciencesJian Jin论文数: 0 引用数: 0 h-index: 0机构: Icahn School of Medicine at Mount Sinai,Mount Sinai Center for Therapeutics Discovery, Department of Pharmacological Sciences
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