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- [1] Design, synthesis and SAR of cyclic boronate-containing macrocyclic inhibitors of HCV NS3/4A serine proteaseABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 239Li, Xianfeng论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAZhang, Yong-Kang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALiu, Yang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USADing, Charles Z.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALi, Qun论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAZhou, Yasheen论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAPlattner, Jacob J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USABaker, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAKraynack, Erica论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAZhang, Suoming论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAFeng, Lisa论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALiu, Liang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAQian, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAFan, Dazhong论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALiao, Liang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAChen, Dianjun论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USANi, Zhi-Jie论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USASlater, Martin J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAJarvest, Richard L.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAThommes, Pia论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAEllis, Malcolm论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAEdge, Colin M.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAHubbard, Julia A.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USANassau, Pam论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAMcDowell, Bill论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USASkarzynski, Tadeusz J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAKazmierski, Wieslaw M.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAWright, Lois L.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USASmith, Gary K.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USACrosby, Renae M.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAWang, Amy A.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAGrimes, Richard M.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USARichardson, Leah论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAWu, Min论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USADong, Xiantao论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALiang, Peng论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAXiao, Jianbin论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALi, Guanghui论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAWang, Shuanghui论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALi, Chong论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USALu, Gang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAZhao, Baojuan论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAZhou, Xinming论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAZou, Wuxin论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAWright, Jon论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAPennicott, Lewis E.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USAPietsch, Inga-Marlene论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA USA
- [2] Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 proteaseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (24) : 7317 - 7322Ding, Charles Z.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhang, Yong-Kang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALi, Xianfeng论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALiu, Yang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhang, Suoming论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhou, Yasheen论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAPlattner, Jacob J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USABaker, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALiu, Liang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USADuan, Maosheng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAJarvest, Richard L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Stevenage SG1 2NY, Herts, England Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAJi, Jingjing论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAKazmierski, Wieslaw M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USATallant, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWright, Lois L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USASmith, Gary K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACrosby, Renae M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWang, Amy A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USANi, Zhi-Jie论文数: 0 引用数: 0 h-index: 0机构: Acme Biosci Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZou, Wuxin论文数: 0 引用数: 0 h-index: 0机构: BioDuro LLC, Beijing 102206, Peoples R China Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWright, Jon论文数: 0 引用数: 0 h-index: 0机构: BioDuro LLC, Beijing 102206, Peoples R China Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA
- [3] Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moietiesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (07) : 2048 - 2054Li, Xianfeng论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhang, Suoming论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhang, Yong-Kang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALiu, Yang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USADing, Charles Z.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhou, Yasheen论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAPlattner, Jacob J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USABaker, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USABu, Wei论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALiu, Liang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAKazmierski, Wieslaw M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USADuan, Maosheng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAGrimes, Richard M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWright, Lois L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USASmith, Gary K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAJarvest, Richard L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Stevenage SG1 2NY, Herts, England Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAJi, Jing-Jing论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACooper, Joel P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USATallant, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACrosby, Renae M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACreech, Katrina论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USANi, Zhi-Jie论文数: 0 引用数: 0 h-index: 0机构: Acme Biosci Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZou, Wuxin论文数: 0 引用数: 0 h-index: 0机构: BioDuro LLC, Beijing 102206, Peoples R China Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWright, Jon论文数: 0 引用数: 0 h-index: 0机构: BioDuro LLC, Beijing 102206, Peoples R China Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA
- [4] IDENTIFICATION OF NOVEL NON-MACROCYCLIC INHIBITORS OF HCV NS3/4A SERINE PROTEASE ACTIVITYHEPATOLOGY, 2008, 48 (04) : 1164A - 1165ABuckman, Brad O.论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAPan, Lin论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAHuang, Lea论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAKossen, Karl论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USARajagopalan, Ravi论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAMisialek, Shawn论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAStevens, Sarah K.论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USATan, Hua论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USARuhrmund, Donald论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USASerebryany, Vladimir论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAMatulik-Adamic, Jasenka论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAStoycheva, Antitsa论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAAmmons, Steve论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USAFuhrer, Douglas K.论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USABlatt, Lawrence M.论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USABeigelman, Leo论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USASeiwert, Scott论文数: 0 引用数: 0 h-index: 0机构: Intermune Inc, Brisbane, CA USA Intermune Inc, Brisbane, CA USA
- [5] Molecular docking study of P4-Benzoxaborole-substituted ligands as inhibitors of HCV NS3/4A proteaseBIOINFORMATION, 2013, 9 (06) : 309 - 314Wadood, Abdul论文数: 0 引用数: 0 h-index: 0机构: Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, Pakistan Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, Pakistan论文数: 引用数: h-index:机构:Jamal, Syed Babar论文数: 0 引用数: 0 h-index: 0机构: Islamic Int Univ, Dept Bioinformat, Islamabad, Pakistan Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, PakistanShah, Masaud论文数: 0 引用数: 0 h-index: 0机构: Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, Pakistan Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, PakistanLodhi, Muhammad Arif论文数: 0 引用数: 0 h-index: 0机构: Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, Pakistan Abdul Wali Khan Univ Mardan, UCS, Dept Biochem, Mardan 23200, Pakistan
- [6] Development of potent macrocyclic inhibitors of genotype 3a HCV NS3/4A proteaseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (23) : 7201 - 7206Rudd, Michael T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcCauley, John A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USARomano, Joseph J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAButcher, John W.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USABush, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcIntyre, Charles J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USANguyen, Kevin T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGilbert, Kevin F.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALyle, Terry A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHolloway, M. Katharine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Chem Modeling & Informat, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAWan, Bang-Lin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAVacca, Joseph P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USASumma, Vincenzo论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, IRBM, Dept Med Chem, Rome, Italy Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHarper, Steven论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, IRBM, Dept Med Chem, Rome, Italy Merck Res Labs, Dept Med Chem, West Point, PA 19486 USARowley, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, IRBM, Dept Med Chem, Rome, Italy Merck Res Labs, Dept Med Chem, West Point, PA 19486 USACarroll, Steven S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USABurlein, Christine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USADiMuzio, Jillian M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGates, Adam论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGraham, Donald J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHuang, Qian论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALudmerer, Steven W.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcClain, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcHale, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAStahlhut, Mark论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAFandozzi, Christine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USATaylor, Anne论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USATrainor, Nicole论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAOlsen, David B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALiverton, Nigel J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA
- [7] Development of macrocyclic inhibitors of HCV NS3/4A protease with cyclic constrained P2-P4 linkersBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (23) : 7207 - 7213Rudd, Michael T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcIntyre, Charles J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USARomano, Joseph J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAButcher, John W.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHolloway, M. Katharine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Chem Modeling & Informat, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USABush, Kimberly论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USANguyen, Kevin T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGilbert, Kevin F.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALyle, Terry A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALiverton, Nigel J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAWan, Bang-Lin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USASumma, Vincenzo论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, IRBM, Dept Med Chem, Rome, Italy Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHarper, Steven论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, IRBM, Dept Med Chem, Rome, Italy Merck Res Labs, Dept Med Chem, West Point, PA 19486 USARowley, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, IRBM, Dept Med Chem, Rome, Italy Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAVacca, Joseph P.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USACarroll, Steven S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USABurlein, Christine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USADiMuzio, Jillian M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGates, Adam论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAGraham, Donald J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAHuang, Qian论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USALudmerer, Steven W.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcClain, Stephanie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcHale, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAStahlhut, Mark论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAFandozzi, Christine论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USATaylor, Anne论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USATrainor, Nicole论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Drug Metab, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAOlsen, David B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Antiviral Res, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USAMcCauley, John A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA Merck Res Labs, Dept Med Chem, West Point, PA 19486 USA
- [8] Novel HCV NS3/4A protease inhibitors with tetrazoyl P* groupsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243Wang, Guoqiang论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USASun, Ying论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USAJiang, Lijuan论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USALu, Xiang论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USAThe-Uyen Phan论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USAChen, Zhigang论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USAMcDaniel, Keith K.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 60064 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USAKempf, Dale J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Abbott Pk, IL 60064 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USAOr, Yat Sun论文数: 0 引用数: 0 h-index: 0机构: Enanta Pharmaceut Inc, Watertown, MA 02472 USA Enanta Pharmaceut Inc, Watertown, MA 02472 USA
- [9] Synthesis and antiviral activity of novel HCV NS3 protease inhibitors with P4 capping groupsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (24) : 7351 - 7356Li, Xianfeng论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALiu, Yang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhang, Yong-Kang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAPlattner, Jacob J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USABaker, Stephen J.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USABu, Wei论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USALiu, Liang论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhou, Yasheen论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USADing, Charles Z.论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAZhang, Suoming论文数: 0 引用数: 0 h-index: 0机构: Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAKazmierski, Wieslaw M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAHamatake, Robert论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USADuan, Maosheng论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWright, Lois L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USASmith, Gary K.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAJarvest, Richard L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Stevenage SG1 2NY, Herts, England Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAJi, Jing-Jing论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACooper, Joel P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USATallant, Matthew D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACrosby, Renae M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USACreech, Katrina论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USAWang, Amy论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Res Triangle Pk, NC 27709 USA Anacor Pharmaceut Inc, Palo Alto, CA 94303 USA
- [10] Treatment of HCV infection with the novel NS3/4A protease inhibitorsCURRENT OPINION IN PHARMACOLOGY, 2014, 18 : 9 - 17De Luca, Andrea论文数: 0 引用数: 0 h-index: 0机构: Univ Senese, Dipartimento Med & Specialist, UOC Malattie Infett Univ, Siena, Italy Univ Cattolica S Cuore, Ist Clin Malattie Infett, Rome, Italy Univ Senese, Dipartimento Med & Specialist, UOC Malattie Infett Univ, Siena, ItalyBianco, Claudia论文数: 0 引用数: 0 h-index: 0机构: Univ Senese, Dipartimento Med & Specialist, UOC Malattie Infett Univ, Siena, Italy Univ Senese, Dipartimento Med & Specialist, UOC Malattie Infett Univ, Siena, ItalyRossetti, Barbara论文数: 0 引用数: 0 h-index: 0机构: Univ Senese, Dipartimento Med & Specialist, UOC Malattie Infett Univ, Siena, Italy Univ Senese, Dipartimento Med & Specialist, UOC Malattie Infett Univ, Siena, Italy