Development of FRET-based receptor conformation sensors for the opioid receptor family and analysis of opioid agonist properties

被引:0
|
作者
Kirchhofer, S. B. [1 ]
Kurz, C. [1 ]
Kurz, M. [1 ]
Buenemann, M. [1 ]
机构
[1] Philipps Univ Marburg, Dept Pharmacol & Clin Pharm, Marburg, Germany
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
P096
引用
收藏
页码:S46 / S46
页数:1
相关论文
共 50 条
  • [1] Dynamics of agonist-evoked opioid receptor activation revealed by FRET- and BRET-based opioid receptor conformation sensors
    Kirchhofer, Sina B.
    Kurz, Claudia
    Geier, Lorenz
    Krett, Anna-Lena
    Krasel, Cornelius
    Buenemann, Moritz
    COMMUNICATIONS BIOLOGY, 2025, 8 (01)
  • [2] Pentapeptides Displaying μ Opioid Receptor Agonist and δ Opioid Receptor Partial Agonist/Antagonist Properties
    Purington, Lauren C.
    Pogozheva, Irina D.
    Traynor, John R.
    Mosberg, Henry I.
    JOURNAL OF MEDICINAL CHEMISTRY, 2009, 52 (23) : 7724 - 7731
  • [3] A comparison of the antinociceptive and adverse effects of a μ-opioid receptor agonist with a δ-opioid receptor agonist
    Gallantine, EL
    Kamali, F
    Meert, TF
    TOXICOLOGY, 2005, 213 (03) : 258 - 258
  • [4] Development of FRET-based sensors for the chemokine receptor CXCR4: Monitoring receptor dynamics and kinetics
    Perpina-Viciano, C.
    Lohse, M. J.
    Hoffmann, C.
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2017, 390 : S25 - S25
  • [5] Development of an efficient and scalable synthesis of a κ-opioid receptor agonist
    Ghosh, A
    Caron, S
    Couturier, M
    DeVries, KM
    Dupont-Gaudet, K
    Hawkins, J
    Ito, F
    Sieser, JE
    Tucker, JL
    Vanderplas, BC
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U3103 - U3104
  • [6] An opioid agonist that does not induce μ-opioid receptor -: Arrestin interactions or receptor internalization
    Groer, C. E.
    Tidgewell, K.
    Moyer, R. A.
    Harding, W. W.
    Rothman, R. B.
    Prisinzano, T. E.
    Bohn, L. M.
    MOLECULAR PHARMACOLOGY, 2007, 71 (02) : 549 - 557
  • [7] FRET-Based Sensors Unravel Activation and Allosteric Modulation of the GABAB Receptor
    Lecat-Guillet, Nathalie
    Monnier, Carine
    Rovira, Xavier
    Kniazeff, Julie
    Lamarque, Laurent
    Zwier, Jurriaan M.
    Trinquet, Eric
    Pin, Jean-Philippe
    Rondard, Philippe
    CELL CHEMICAL BIOLOGY, 2017, 24 (03): : 360 - 370
  • [8] Development of bifunctional mu opioid receptor (MOR) agonist/delta opioid receptor (DOR) antagonist peptides and peptidomimetics
    Mosberg, Henry I.
    Anand, Jessica
    Bender, Aaron
    Harland, Aubrie A.
    Sobczyk-Kojiro, Katarzyna
    Yeomans, Larisa
    Jutkiewicz, Emily M.
    Traynor, John
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248
  • [9] Research and development of κ opioid receptor agonists and δ opioid receptor agonists
    Nagase, Hiroshi
    Saitoh, Akiyoshi
    PHARMACOLOGY & THERAPEUTICS, 2020, 205
  • [10] Differential opioid agonist regulation of the mouse mu opioid receptor
    Blake, AD
    Bot, G
    Freeman, JC
    Reisine, T
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1997, 272 (02) : 782 - 790