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- [1] A multi-center, open-label, randomized dose expansion study of PF-06821497, a potent and selective inhibitor of enhancer of zeste homolog 2 (EZH2), in patients with metastatic castration-resistant prostate cancer (mCRPC).JOURNAL OF CLINICAL ONCOLOGY, 2023, 41Calvo, Mariona论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainPenkov, Konstantin论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainSpira, Alexander I.论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainCandilejo, Irene Moreno论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainShore, Neal D.论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainZhang, Tian论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainMellado-Gonzalez, Begona论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainGordoa, Teresa Alonso论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainRodriguez, Luis Paz-Ares论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainTarantolo, Stefano R.论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainSoto, Juan Jose论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainAlter, Robert S.论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainAndreu-Vieyra, Claudia论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainBowler, Timothy论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainMaity, Arnab K.论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainHariharan, Subramanian论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, SpainSchweizer, Michael Thomas论文数: 0 引用数: 0 h-index: 0机构: Catalan Inst Oncol, Hosp, Med Oncol Dept, Barcelona, Spain
- [2] Phase 1 trial of mevrometostat (PF-06821497), a potent and selective inhibitor of enhancer of zeste homolog 2 (EZH2), in castration-resistant prostate cancer (CRPC).JOURNAL OF CLINICAL ONCOLOGY, 2024, 42 (16)Schweizer, Michael Thomas论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USAPenkov, Konstantin论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USAChoudhury, Atish Dipankar论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USACalvo, Emiliano论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USAFrank, Richard C.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USALiu, Li论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USAMittapalli, Rajendar K.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USATougias, Jessica论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USAAndreu-Vieyra, Claudia论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USABowler, Timothy Geoffrey论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USASoman, Neelesh论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USAGarmezy, Benjamin论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA 98195 USA
- [3] Phase I trial of PF-06821497, a potent and selective inhibitor of enhancer of zeste homolog 2 (EZH2), in follicular lymphoma (FL), small cell lung cancer (SCLC) and castration-resistant prostate cancer (CRPC)ANNALS OF ONCOLOGY, 2022, 33 (07) : S763 - S764Schweizer, M.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Div Med Oncol, Seattle, WA USA Univ Washington, Div Med Oncol, Seattle, WA USAPenkov, K. D.论文数: 0 引用数: 0 h-index: 0机构: Private Med Inst Euromedserv, Gen Dept, St Petersburg, Russia Univ Washington, Div Med Oncol, Seattle, WA USATolcher, A. W.论文数: 0 引用数: 0 h-index: 0机构: NEXT Oncol, Clin Res, San Antonio, TX USA Univ Washington, Div Med Oncol, Seattle, WA USAChoudhury, A. D.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Prostate Canc Ctr, Boston, MA USA Univ Washington, Div Med Oncol, Seattle, WA USADoronin, V.论文数: 0 引用数: 0 h-index: 0机构: Moscow City Clin Hosp 40, State Budgetary Healthcare Inst, Clin Hosp, Moscow, Russia Univ Washington, Div Med Oncol, Seattle, WA USAAljumaily, R.论文数: 0 引用数: 0 h-index: 0机构: Univ Oklahoma, Stephenson Canc Ctr, Div Hematol Oncol, Oklahoma City, OK USA Univ Washington, Div Med Oncol, Seattle, WA USACalvo, E.论文数: 0 引用数: 0 h-index: 0机构: START Madrid Grp, Med Oncol, Madrid, Spain Univ Washington, Div Med Oncol, Seattle, WA USAFrank, R. C.论文数: 0 引用数: 0 h-index: 0机构: Nuvance Hlth, Norwalk Hosp, Dept Med, Norwalk, CT USA Univ Washington, Div Med Oncol, Seattle, WA USAHamm, J. T.论文数: 0 引用数: 0 h-index: 0机构: Norton Canc Inst, Med Oncol Dept, Louisville, KY USA Univ Washington, Div Med Oncol, Seattle, WA USAGarcia, V. Moreno论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ Fdn Jimenez Diaz, START Madrid FJD, Early Phase Clin Trials Unit, Madrid, Spain Univ Washington, Div Med Oncol, Seattle, WA USAVorobyev, V.论文数: 0 引用数: 0 h-index: 0机构: Botkin Hosp, Bone Marrow Transplant Dept, Moscow, Russia Univ Washington, Div Med Oncol, Seattle, WA USABillotte, S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Canc Vaccines, San Diego, CA USA Univ Washington, Div Med Oncol, Seattle, WA USABowler, T.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Clin, New York, NY USA Univ Washington, Div Med Oncol, Seattle, WA USAChen, J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc USA, Global Prod Dev Oncol, San Francisco, CA USA Univ Washington, Div Med Oncol, Seattle, WA USALin, T.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Clin Dev, New York, NY USA Univ Washington, Div Med Oncol, Seattle, WA USALiu, L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, La Jolla Campus CB10, San Diego, CA USA Univ Washington, Div Med Oncol, Seattle, WA USAMaity, A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Oncol Clin Trials, San Diego, CA USA Univ Washington, Div Med Oncol, Seattle, WA USASharma, S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer, Sci, San Diego, CA USA Univ Washington, Div Med Oncol, Seattle, WA USAJohnson, M. L.论文数: 0 引用数: 0 h-index: 0机构: Tennessee Oncol PLLC, Sarah Cannon Res Inst, Med Oncol, Nashville, TN USA Univ Washington, Div Med Oncol, Seattle, WA USA
- [4] Inhibition of enhancer of zeste homolog 2 (EZH2) overcomes enzalutamide resistance in castration-resistant prostate cancerJOURNAL OF BIOLOGICAL CHEMISTRY, 2019, 294 (25) : 9911 - 9923Bai, Yunfeng论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA Shanxi Datong Univ, Sch Chem & Environm Engn, Datong 037009, Shanxi, Peoples R China Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USAZhang, Zhuangzhuang论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USACheng, Lijun论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Biomed Informat, Columbus, OH 43210 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USAWang, Ruixin论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USAChen, Xiaoliang论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA Shanxi Datong Univ, Sch Chem & Environm Engn, Datong 037009, Shanxi, Peoples R China Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USAKong, Yifan论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USAFeng, Feng论文数: 0 引用数: 0 h-index: 0机构: Shanxi Datong Univ, Sch Chem & Environm Engn, Datong 037009, Shanxi, Peoples R China Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USAAhmad, Nihal论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Dept Dermatol, Madison, WI 53715 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USALi, Lang论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Dept Biomed Informat, Columbus, OH 43210 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USALiu, Xiaoqi论文数: 0 引用数: 0 h-index: 0机构: Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA Univ Kentucky, Markey Canc Ctr, Lexington, KY 40536 USA Univ Kentucky, Dept Toxicol & Canc Biol, Lexington, KY 40536 USA
- [5] Discovery of a novel class of potent, selective, and orally bioavailable histone methyltransferase Enhancer of Zeste Homolog 2 (EZH2) inhibitors and the identification of development candidate PF-06821497ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253Kung, Pei-Pei论文数: 0 引用数: 0 h-index: 0机构: Pfizer WRD La Jolla, San Diego, CA USA Pfizer WRD La Jolla, San Diego, CA USABergqvist, Simon论文数: 0 引用数: 0 h-index: 0机构: Pfizer WRD La Jolla, San Diego, CA USABingham, Patrick论文数: 0 引用数: 0 h-index: 0机构: Pfizer WRD La Jolla, San Diego, CA USA Pfizer WRD La Jolla, San Diego, CA USABraganza, John论文数: 0 引用数: 0 h-index: 0机构: Pfizer WRD La Jolla, San Diego, CA USA Pfizer WRD La Jolla, San Diego, CA USABrooun, Alexei论文数: 0 引用数: 0 h-index: 0机构: Pfizer WRD La Jolla, San Diego, CA USA Pfizer WRD La Jolla, San Diego, CA USACollins, Michael论文数: 0 引用数: 0 h-index: 0机构: Pfizer WRD La Jolla, San Diego, CA USA Pfizer WRD La Jolla, San Diego, CA USADiehl, Wade论文数: 0 引用数: 0 h-index: 0机构: Pfizer 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- [6] Enhancer of zeste-homolog 2 (EZH2) expression and clinical outcomes in metastatic castrate resistant prostate cancer (mCRPC).JOURNAL OF CLINICAL ONCOLOGY, 2018, 36 (06)Giridhar, Karthik论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USACostello, Brian Addis论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USASosa, Carlos论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USAHuang, Haojie论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USAKohli, Manish论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA
- [7] A phase 1/2, open-label, randomized, dose-finding and dose expansion study of gedatolisib in combination with darolutamide in metastatic castration-resistant prostate cancer (mCRPC)CANCER RESEARCH, 2024, 84 (07)Sharp, Adam论文数: 0 引用数: 0 h-index: 0Bernard-Tessier, Alice论文数: 0 引用数: 0 h-index: 0Borchiellini, Delphine论文数: 0 引用数: 0 h-index: 0de Bono, Johann论文数: 0 引用数: 0 h-index: 0Fizazi, Karim论文数: 0 引用数: 0 h-index: 0Gravis, Gwenaelle论文数: 0 引用数: 0 h-index: 0Lorente, David论文数: 0 引用数: 0 h-index: 0Mahammedi, Hakim论文数: 0 引用数: 0 h-index: 0Mellado, Begona论文数: 0 引用数: 0 h-index: 0Olmos, David论文数: 0 引用数: 0 h-index: 0Pacey, Simon论文数: 0 引用数: 0 h-index: 0Piulats, Jose论文数: 0 引用数: 0 h-index: 0Ramirez, Sara P.论文数: 0 引用数: 0 h-index: 0Gorbatchevsky, Igor论文数: 0 引用数: 0 h-index: 0Heath, Elisabeth论文数: 0 引用数: 0 h-index: 0
- [8] A phase 1/2, open-label, randomized, dose-finding and dose expansion study of gedatolisib in combination with darolutamide in metastatic castration-resistant prostate cancer (mCRPC)JOURNAL OF CLINICAL ONCOLOGY, 2024, 42 (16)Heath, Elisabeth I.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USASharp, Adam论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USABorchiellini, Delphine论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USADe Bono, Johann S.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAFizazi, Karim论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAGravis, Gwenaelle论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USALorente, David论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAMahammedi, Hakim论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAMellado-Gonzalez, Bego Na论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAOlmos, David论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAPacey, Simon论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAPiulats, Josep M.论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USARamirez, Sara Perez论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USAGorbatchevsky, Igor论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USABernard-Tessier, Alice论文数: 0 引用数: 0 h-index: 0机构: Wayne State Univ, Barbara Ann Karmanos Canc Inst, Dept Oncol, Sch Med, Detroit, MI USA
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