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- [1] RAS:RAF proximity ligation assay may predict response to KRASG12C inhibitors in NSCLCMOLECULAR CANCER RESEARCH, 2023, 21 (05)Kato, Ryoji论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USASolanki, Hitendra S.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USAImbody, Denis论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USAMajumder, Anurima论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USAStern, Yaakov论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USABridenstine, Liznair论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USAJohnson, Joseph论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USAHaura, Eric B.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA
- [2] In Situ RAS:RAF Binding Correlates with Response to KRASG12C Inhibitors in KRASG12C-Mutant Non-Small Cell Lung CancerCLINICAL CANCER RESEARCH, 2025, 31 (06) : 1150 - 1162Kato, Ryoji论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USASolanki, Hitendra S.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAOzakinci, Hilal论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USADesai, Bina论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Metab & Physiol, Tampa, FL USA Univ S Florida, Canc Biol Ph D Program, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAGundlapalli, Harika论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Translat Sci, Redwood City, CA USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAYang, Yu Chi论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Translat Sci, Redwood City, CA USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAAronchik, Ida论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Translat Sci, Redwood City, CA USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USASingh, Mallika论文数: 0 引用数: 0 h-index: 0机构: Revolut Med, Translat Sci, Redwood City, CA USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAJohnson, Joseph论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Analyt Microscopy Core Facil, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAMarusyk, Andriy论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Metab & Physiol, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USABoyle, Theresa A.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Pathol, Tampa, FL USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USAHaura, Eric B.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USA H Lee Moffitt Canc Ctr & Res Inst, Dept Thorac Oncol, 12902 Magnolia Dr, Tampa, FL 33612 USA
- [3] TEAD Inhibitors Sensitize KRASG12C Inhibitors via Dual Cell Cycle Arrest in KRASG12C-Mutant NSCLCPHARMACEUTICALS, 2023, 16 (04)Tammaccaro, Salvina Laura论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FrancePrigent, Philippe论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceLe Bail, Jean-Christophe论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceDos-Santos, Odette论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceDassencourt, Laurent论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceEskandar, Myriam论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceBuzy, Armelle论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Bio Struct & Biophys, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceVenier, Olivier论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Small Mol Med Chem, F-91380 Chilly Mazarin, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceGuillemot, Jean-Claude论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Genom & Prote, Translat Sci, F-91380 Chilly Mazarin, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceVeeranagouda, Yaligara论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Genom & Prote, Translat Sci, F-91380 Chilly Mazarin, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceDidier, Michel论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Genom & Prote, Translat Sci, F-91380 Chilly Mazarin, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceSpanakis, Emmanuel论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Precis Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceKanno, Tokuwa论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Precis Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceCesaroni, Matteo论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Precis Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceMathieu, Stephane论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Mol & Digital Histopathol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceCanard, Luc论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Mol & Digital Histopathol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceCasse, Alhassan论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Mol & Digital Histopathol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceWindenberger, Fanny论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Nonclin Efficacy & Safety, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceCalvet, Loreley论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Pharmacol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceNoblet, Laurence论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Pharmacol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceSidhu, Sukhvinder论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Pharmacol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceDebussche, Laurent论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceMoll, Jurgen论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, FranceValtingojer, Iris论文数: 0 引用数: 0 h-index: 0机构: Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France Sanofi R&D, Oncol, F-94400 Vitry Sur Seine, France
- [4] Development of a biotin-streptavidin-enhanced enzyme-linked immunosorbent assay (BA-ELISA) for high-throughput screening of KRASG12C inhibitorsSLAS DISCOVERY, 2022, 27 (02) : 107 - 113Liu, Shuang论文数: 0 引用数: 0 h-index: 0机构: Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R China Shouyao Holdings Beijing Co Ltd, Discovery Biol Dept, Beijing 100195, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R ChinaShi, Junfen论文数: 0 引用数: 0 h-index: 0机构: Shouyao Holdings Beijing Co Ltd, Discovery Biol Dept, Beijing 100195, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R ChinaLi, Hongjuan论文数: 0 引用数: 0 h-index: 0机构: Shouyao Holdings Beijing Co Ltd, Discovery Biol Dept, Beijing 100195, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R ChinaLi, Jijun论文数: 0 引用数: 0 h-index: 0机构: Shouyao Holdings Beijing Co Ltd, Med Chem Dept, Beijing, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R ChinaZhu, Yan论文数: 0 引用数: 0 h-index: 0机构: Shouyao Holdings Beijing Co Ltd, Med Chem Dept, Beijing, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R ChinaLi, Binghui论文数: 0 引用数: 0 h-index: 0机构: Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R ChinaSun, Yinghui论文数: 0 引用数: 0 h-index: 0机构: Shouyao Holdings Beijing Co Ltd, Discovery Biol Dept, Beijing 100195, Peoples R China Capital Med Univ, Dept Biochem & Mol Biol, Beijing 100069, Peoples R China
- [5] De Novo Rational design of peptide-based covalent inhibitors via mapping of complementary binding site residues – technical protocol and case study on KRASG12C and BTK481CBMC Methods, 2 (1):Ernest Oduro-Kwateng论文数: 0 引用数: 0 h-index: 0机构: University of KwaZulu Natal,Molecular Bio University of KwaZulu Natal,Molecular BioMusab Ali论文数: 0 引用数: 0 h-index: 0机构: University of KwaZulu Natal,Molecular Bio University of KwaZulu Natal,Molecular BioIbrahim Oluwatobi Kehinde论文数: 0 引用数: 0 h-index: 0机构: University of KwaZulu Natal,Molecular Bio University of KwaZulu Natal,Molecular BioLi Rao论文数: 0 引用数: 0 h-index: 0机构: Central China Normal University,Computation and Drug Design Research Group, School of Health Sciences University of KwaZulu Natal,Molecular BioMahmoud E. S. Soliman论文数: 0 引用数: 0 h-index: 0机构: University of KwaZulu Natal,Molecular Bio University of KwaZulu Natal,Molecular Bio