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- [1] Preliminary analysis of pharmacokinetic (PK) and target engagement biomarkers from a first in human phase 1 study of immunomodulatory aryl hydrocarbon receptor (AhR) inhibitor BAY2416964CANCER RESEARCH, 2023, 83 (08)Papadopoulos, Kyriakos论文数: 0 引用数: 0 h-index: 0Cecchini, Michael论文数: 0 引用数: 0 h-index: 0Lopez, Juanita S.论文数: 0 引用数: 0 h-index: 0Jager, Dirk论文数: 0 引用数: 0 h-index: 0Chung, Ki Young论文数: 0 引用数: 0 h-index: 0Platten, Michael论文数: 0 引用数: 0 h-index: 0Prinz, Florian论文数: 0 引用数: 0 h-index: 0Ishii, Yuko论文数: 0 引用数: 0 h-index: 0Schaer, David论文数: 0 引用数: 0 h-index: 0Gutcher, Ilona论文数: 0 引用数: 0 h-index: 0Leder, Gabriele论文数: 0 引用数: 0 h-index: 0Pencheva, Radost论文数: 0 引用数: 0 h-index: 0Wagener, Thomas论文数: 0 引用数: 0 h-index: 0Scheerans, Christian论文数: 0 引用数: 0 h-index: 0Zieschang, Carsten论文数: 0 引用数: 0 h-index: 0Wagner, Andrea论文数: 0 引用数: 0 h-index: 0Stamatelos, Spyros论文数: 0 引用数: 0 h-index: 0Dumbrava, Ecaterina论文数: 0 引用数: 0 h-index: 0
- [2] First-in-human phase I study of the microtubule inhibitor plocabulin in patients with advanced solid tumorsInvestigational New Drugs, 2019, 37 : 674 - 683Elena Elez论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Carlos Gomez-Roca论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Arturo Soto Matos-Pita论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Guillem Argiles论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Thibaud Valentin论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Cinthya Coronado论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Jorge Iglesias论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Teresa Macarulla论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Sarah Betrian论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Salvador Fudio论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Katrin Zaragoza论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Josep Tabernero论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)Jean-Pierre Delord论文数: 0 引用数: 0 h-index: 0机构: Universitat Autònoma de Barcelona,Vall d’Hebron University Hospital and Vall d’Hebron Institute of Oncology (VHIO)
- [3] First-in-human phase I study of the microtubule inhibitor plocabulin in patients with advanced solid tumorsINVESTIGATIONAL NEW DRUGS, 2019, 37 (04) : 674 - 683Elez, Elena论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, Spain Univ Autonoma Barcelona, VHIO, Barcelona, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainGomez-Roca, Carlos论文数: 0 引用数: 0 h-index: 0机构: IUCT Oncopole, Inst Claudius Regaud, Clin Res Unit, 1 Ave Joliot Curie, F-31059 Toulouse, France Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainSoto Matos-Pita, Arturo论文数: 0 引用数: 0 h-index: 0机构: Pharma Mar SA, Clin R&D, Madrid, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainArgiles, Guillem论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, Spain Univ Autonoma Barcelona, VHIO, Barcelona, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainValentin, Thibaud论文数: 0 引用数: 0 h-index: 0机构: IUCT Oncopole, Inst Claudius Regaud, Clin Res Unit, 1 Ave Joliot Curie, F-31059 Toulouse, France Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainCoronado, Cinthya论文数: 0 引用数: 0 h-index: 0机构: Pharma Mar SA, Clin R&D, Madrid, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainIglesias, Jorge论文数: 0 引用数: 0 h-index: 0机构: Pharma Mar SA, Clin R&D, Madrid, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainMacarulla, Teresa论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, Spain Univ Autonoma Barcelona, VHIO, Barcelona, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainBetrian, Sarah论文数: 0 引用数: 0 h-index: 0机构: IUCT Oncopole, Inst Claudius Regaud, Clin Res Unit, 1 Ave Joliot Curie, F-31059 Toulouse, France Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainFudio, Salvador论文数: 0 引用数: 0 h-index: 0机构: Pharma Mar SA, Clin R&D, Madrid, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainZaragoza, Katrin论文数: 0 引用数: 0 h-index: 0机构: Pharma Mar SA, Clin R&D, Madrid, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainTabernero, Josep论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, Spain Univ Autonoma Barcelona, VHIO, Barcelona, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, SpainDelord, Jean-Pierre论文数: 0 引用数: 0 h-index: 0机构: IUCT Oncopole, Inst Claudius Regaud, Clin Res Unit, 1 Ave Joliot Curie, F-31059 Toulouse, France Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona, Spain
- [4] RESULTS OF A FIRST-IN-HUMAN PHASE I STUDY OF THE ALK INHIBITOR LDK378 IN ADVANCED SOLID TUMORSANNALS OF ONCOLOGY, 2012, 23 : 153 - 153Shaw, A. T.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Boston, MA USA Harvard Univ, Sch Med, Boston, MA USACamidge, D. R.论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Sch Med, Denver, CO USA Harvard Univ, Sch Med, Boston, MA USAFelip, E.论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Univ Hosp, Barcelona, Spain Harvard Univ, Sch Med, Boston, MA USASharma, S.论文数: 0 引用数: 0 h-index: 0机构: Ctr Invest Therapeut, Huntsman Canc Inst, Salt Lake City, UT USA Harvard Univ, Sch Med, Boston, MA USATan, D. S. W.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Dept Med Oncol, Singapore, Singapore Harvard Univ, Sch Med, Boston, MA USAKim, D.论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ Hosp, Dept Internal Med, Seoul 110744, South Korea Harvard Univ, Sch Med, Boston, MA USADe Pas, T.论文数: 0 引用数: 0 h-index: 0机构: Ist Europeo Oncol, Med Oncol Unit Resp Tract & Sarcomas, Milan, Italy Harvard Univ, Sch Med, Boston, MA USAVansteenkiste, J. F.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Gasthuisberg, Resp Oncol Unit Pulmonol, B-3000 Louvain, Belgium Harvard Univ, Sch Med, Boston, MA USASantoro, A.论文数: 0 引用数: 0 h-index: 0机构: Ist Clin Humanitas, Dept Med Oncol & Hematol, Rozzano, Italy Harvard Univ, Sch Med, Boston, MA USALiu, G.论文数: 0 引用数: 0 h-index: 0机构: Princess Margeret Hosp, Ontario Canc Inst, Toronto, ON, Canada Harvard Univ, Sch Med, Boston, MA USAGoldwasser, M.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, Novartis Inst BioMed Res, Cambridge, MA USA Harvard Univ, Sch Med, Boston, MA USADai, D.论文数: 0 引用数: 0 h-index: 0机构: Novartis Pharmaceut, Oncol Clin Pharmacol, E Hanover, NJ USA Harvard Univ, Sch Med, Boston, MA USABoral, A. L.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res Inc, Clin Res, Cambridge, MA USA Harvard Univ, Sch Med, Boston, MA USAMehra, R.论文数: 0 引用数: 0 h-index: 0机构: Fox Chase Canc Ctr, Dept Dev Therapeut, Philadelphia, PA 19111 USA Harvard Univ, Sch Med, Boston, MA USA
- [5] A first-in-human phase I study of TAS-117, an allosteric AKT inhibitor, in patients with advanced solid tumorsCANCER CHEMOTHERAPY AND PHARMACOLOGY, 2024, 93 (06) : 605 - 616Doi, Toshihiko论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanTakahashi, Shunji论文数: 0 引用数: 0 h-index: 0机构: Canc Inst Hosp, Japanese Fdn Canc Res, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanAoki, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Keio Univ, Sch Med, Tokyo, Japan Akasaka Sannou Med Ctr, Tokyo, Japan Int Univ Hlth & Welf, Grad Sch, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanYonemori, Kan论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHara, Hiroki论文数: 0 引用数: 0 h-index: 0机构: Saitama Canc Ctr, Kita Adachi, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHasegawa, Kosei论文数: 0 引用数: 0 h-index: 0机构: Saitama Med Univ, Int Med Ctr, Hidaka, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanTakehara, Kazuhiro论文数: 0 引用数: 0 h-index: 0机构: NHO Shikoku Canc Ctr, Matsuyama, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHarano, Kenichi论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Hosp East, Kashiwa, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanYunokawa, Mayu论文数: 0 引用数: 0 h-index: 0机构: Canc Inst Hosp, Japanese Fdn Canc Res, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, Japan论文数: 引用数: h-index:机构:Shimoi, Tatsunori论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr, Tokyo, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanHorie, Koji论文数: 0 引用数: 0 h-index: 0机构: Saitama Canc Ctr, Kita Adachi, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanOgasawara, Aiko论文数: 0 引用数: 0 h-index: 0机构: Saitama Med Univ, Int Med Ctr, Hidaka, Japan Natl Canc Ctr Hosp East, Kashiwa, JapanOkame, Shinichi论文数: 0 引用数: 0 h-index: 0机构: NHO Shikoku Canc Ctr, Matsuyama, Japan Natl Canc Ctr Hosp East, Kashiwa, Japan
- [6] A Phase I First-in-Human Pharmacokinetic and Pharmacodynamic Study of Serdemetan in Patients with Advanced Solid TumorsCLINICAL CANCER RESEARCH, 2011, 17 (19) : 6313 - 6321Tabernero, Josep论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainDirix, Luc论文数: 0 引用数: 0 h-index: 0机构: Sint Augustinus, Antwerp, Belgium Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainSchoffski, Patrick论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Leuven, Dept Gen Med Oncol, Louvain, Belgium Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainCervantes, Andres论文数: 0 引用数: 0 h-index: 0机构: Univ Valencia, INCLIVA, Hosp Clin, Dept Hematol & Med Oncol, Valencia, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainAntonio Lopez-Martin, Jose论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ 12 Octubre, Madrid, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainCapdevila, Jaume论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, Spain Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, Spainvan Beijsterveldt, Ludy论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Raritan, NJ USA Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainPlatero, Suso论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Raritan, NJ USA Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainHall, Brett论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Raritan, NJ USA Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainYuan, Zhilong论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Raritan, NJ USA Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainKnoblauch, Roland论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Raritan, NJ USA Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, SpainZhuang, Sen Hong论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev LLC, Raritan, NJ USA Univ Autonoma Barcelona, Vall dHebron Univ Hosp, Barcelona 08035, Spain
- [7] Updated results from a phase I, open-label, multicenter, first-in-human study of AMG 404, a checkpoint inhibitor, in patients with advanced solid tumorsANNALS OF ONCOLOGY, 2021, 32 : S1440 - S1442Price, T. J.论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, Australia Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaPrenen, H.论文数: 0 引用数: 0 h-index: 0机构: UZA, Univ Antwerp Hosp, Oncol Dept, Edegem, Belgium Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaLugowska, I.论文数: 0 引用数: 0 h-index: 0机构: Maria Sklodowska Curie Natl Res Inst Oncol, Dept Soft Tissue Bone Sarcoma & Melanoma MSCMI, Warsaw, Poland Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaFalchook, G. S.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Drug Dev, New York, NY USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaMonzon, J. G.论文数: 0 引用数: 0 h-index: 0机构: Tom Baker Canc Clin, Med Oncol, Calgary, AB, Canada Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaArkenau, H. T.论文数: 0 引用数: 0 h-index: 0机构: SCRI, Sarah Cannon Res Inst SCRI UK, London, England Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaChawla, S. P.论文数: 0 引用数: 0 h-index: 0机构: Sarcoma Oncol Res Ctr, Oncol, Santa Monica, CA USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaHui, M. N.论文数: 0 引用数: 0 h-index: 0机构: Chris OBrien Lifehouse, Med Oncol, Camperdown, NSW, Australia Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaKuboki, Y.论文数: 0 引用数: 0 h-index: 0机构: Hosp East, Natl Canc Ctr, Expt Therapeut & GI Oncol Dept, Kashiwa, Chiba, Japan Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaDziadziuszko, R.论文数: 0 引用数: 0 h-index: 0机构: Med Univ Gdansk, Oncol & Radiotherapy Dept, Gdansk, Poland Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaOzawa, Y.论文数: 0 引用数: 0 h-index: 0机构: Wakayama Med Univ, Internal Med Dept 3, Wakayama, Japan Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaFernandez, M. E. Elez论文数: 0 引用数: 0 h-index: 0机构: Vall dHebron Univ Hosp, Med Oncol Dept, Barcelona, Spain Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaLima, C. S. P. Rocha论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ, Ctr Comprehens Canc, Div Hematol & Oncol, Winston Salem, NC 27101 USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaSubbiah, V.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Invest Canc Therapeut, Houston, TX 77030 USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaTan, D. S. W.论文数: 0 引用数: 0 h-index: 0机构: Natl Canc Ctr Singapore, NCCS, Med Oncol, Singapore, Singapore Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaWang, K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Biostat, Thousand Oaks, CA 91320 USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaHindoyan, A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Biomarkers, Thousand Oaks, CA 91320 USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaShi, W.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Biomarkers, San Francisco, CA USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaKistler, M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Clin Dev, Thousand Oaks, CA 91320 USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, AustraliaSadraei, N. Hashemi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Clin Dev, Thousand Oaks, CA 91320 USA Queen Elizabeth Hosp, Emergency Dept, Med Oncol, Woodville, SA, Australia
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