Synthesis of Novel Ligustrazine Derivatives as Potential Platelet Aggregation Inhibitors

被引：0

作者：

Xian Chao CHENG

机构：

来源：

Chinese Chemical Letters | 2006年 / 10期

关键词：

Synthesis; ligustrazine; derivatives; platelet aggregation inhibitors;

D O I：

暂无

中图分类号：

O621.3 [有机合成化学];

学科分类号：

070303 ; 081704 ;

摘要：

A series of novel ligustrazine derivatives were synthesized. These compounds have not been reported in literature, and their chemical structures were confirmed by IR, 1H NMR and ESI-MS. The preliminary antiplatelet aggregation screening results demonstrated that the compounds 7a, 7b and 7c showed higher potency than ligustrazine.

引用

页码：1317 / 1320

页数：4

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