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- [1] The novel potent TEAD inhibitor, K-975, inhibits YAP1/TAZ-TEAD protein-protein interactions and exerts an anti-tumor effect on malignant pleural mesotheliomaAMERICAN JOURNAL OF CANCER RESEARCH, 2020, 10 (12): : 4399 - 4415Kaneda, Ayumi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Tokyo Inst Technol, Sch Life Sci & Technol, Yokohama, Kanagawa, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanSeike, Toshihiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanDanjo, Tomohiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanNakajima, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanOtsubo, Nobumasa论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanYamaguchi, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanTsuji, Yoshiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanHamaguchi, Kaori论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanYasunaga, Mai论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanNishiya, Yoichi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanSuzuki, Michihiko论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanSaito, Jun-ichi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanYatsunami, Rie论文数: 0 引用数: 0 h-index: 0机构: Tokyo Inst Technol, Sch Life Sci & Technol, Yokohama, Kanagawa, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanNakamura, Satoshi论文数: 0 引用数: 0 h-index: 0机构: Tokyo Inst Technol, Sch Life Sci & Technol, Yokohama, Kanagawa, Japan Numazu Coll, Natl Inst Technol, Shizuoka, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanSekido, Yoshitaka论文数: 0 引用数: 0 h-index: 0机构: Aichi Canc Ctr Res Inst, Div Canc Biol, Nagoya, Aichi, Japan Nagoya Univ, Div Mol & Cellular Oncol, Grad Sch Med, Nagoya, Aichi, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, JapanMori, Kiyotoshi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan Kyowa Kirin Co Ltd, R&D Div, 1188 Shimotogari,Nagaizumi Cho, Shizuoka 4118731, Japan
- [2] OPN-9840, a non-covalent potent pan-TEAD inhibitor, exhibits single agent efficacy in preclinical malignant mesothelioma modelsCANCER RESEARCH, 2024, 84 (06)Chen, Pan-Yu论文数: 0 引用数: 0 h-index: 0Matusow, Bernice论文数: 0 引用数: 0 h-index: 0Tsai, James论文数: 0 引用数: 0 h-index: 0Li, Peipei论文数: 0 引用数: 0 h-index: 0Hoa Nguyen论文数: 0 引用数: 0 h-index: 0Habets, Gaston论文数: 0 引用数: 0 h-index: 0Bollag, Gideon论文数: 0 引用数: 0 h-index: 0Chowdhury, Somenath论文数: 0 引用数: 0 h-index: 0
- [3] Discovery of a first-in-class TEAD inhibitor which directly inhibits YAP/TAZ-TEAD protein-protein interaction and shows a potent anti-tumor effect in malignant pleural mesotheliomaCANCER RESEARCH, 2019, 79 (13)Kaneda, Ayumi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanSeike, Toshihiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanUemori, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanMyojo, Kensuke论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanAida, Kensuke论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanDanjo, Tomohiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanNakajima, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanYamaguchi, Daisuke论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanHamada, Tomoko论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanTsuji, Yoshiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanHamaguchi, Kaori论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanYasunaga, Mai论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanOtsubo, Nobumasa论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanOnodera, Hideyuki论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanNishiya, Yoichi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanSuzuki, Michihiko论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanSaito, Junichi论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanIshii, Toshihiko论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, JapanNakai, Ryuichiro论文数: 0 引用数: 0 h-index: 0机构: Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan Kyowa Hakko Kirin Co Ltd, Nagaizumi, Shizuoka, Japan
- [4] ISM6331, a novel and potent pan-TEAD inhibitor, exhibits strong antitumor activity in preclinical models of Hippo pathway-dysregulated cancersCANCER RESEARCH, 2024, 84 (06)Li, Qi论文数: 0 引用数: 0 h-index: 0Wan, Jainfei论文数: 0 引用数: 0 h-index: 0Liu, Jinxin论文数: 0 引用数: 0 h-index: 0Shang, Jing论文数: 0 引用数: 0 h-index: 0Yu, Jiaojiao论文数: 0 引用数: 0 h-index: 0Zhu, Wei论文数: 0 引用数: 0 h-index: 0Chen, Celia X. -J.论文数: 0 引用数: 0 h-index: 0Qiao, Junwen论文数: 0 引用数: 0 h-index: 0Wang, Ling论文数: 0 引用数: 0 h-index: 0Zhang, Man论文数: 0 引用数: 0 h-index: 0Ding, Xiao论文数: 0 引用数: 0 h-index: 0Bavadekar, Supriya论文数: 0 引用数: 0 h-index: 0Rao, Sujata论文数: 0 引用数: 0 h-index: 0Ren, Feng论文数: 0 引用数: 0 h-index: 0Zhavoronkov, Alex论文数: 0 引用数: 0 h-index: 0