Design, Synthesis, and Anti-Alzheimer Activity of 2,5-Disubstituted 1,3,4-Thiadiazole: Kinetic Studies, Molecular Docking, and MD Simulations

被引:0
|
作者
M. L. Sujatha [1 ]
Prabhu Jalihal [2 ]
Manjunatha S. Katagi [3 ]
Durgesh Paresh Bidye [4 ]
Sheshagiri R. Dixit [4 ]
B. P. Nandeshwarappa [1 ]
机构
[1] Department of Studies in Chemistry,
[2] Davangere University,undefined
[3] Shivagangotri,undefined
[4] Davangere,undefined
[5] Department of Pharmaceutical Chemistry,undefined
[6] HSK College of Pharmacy,undefined
[7] Bagalkot,undefined
[8] Department of Pharmaceutical Chemistry,undefined
[9] Bapuji Pharmacy College,undefined
[10] Davangere,undefined
[11] Department of Pharmaceutical Chemistry,undefined
[12] JSS College of Pharmacy,undefined
[13] SS Nagar,undefined
[14] Mysore,undefined
[15] JSS Academy of Higher Education and Research,undefined
关键词
acetylcholinesterase; Alzheimer’s disease; 1,3,4-thiadiazole; antioxidant activity; Ellman’s method;
D O I
10.1134/S1068162024605858
中图分类号
学科分类号
摘要
引用
收藏
页码:912 / 931
页数:19
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