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- [4] THE GABRIEL-COLMAN REARRANGEMENT IN BIOLOGICAL-SYSTEMS - DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF PHTHALIMIDE AND SACCHARIN DERIVATIVES AS POTENTIAL MECHANISM-BASED INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, CATHEPSIN-G AND PROTEINASE-3 BIOORGANIC & MEDICINAL CHEMISTRY, 1995, 3 (02) : 187 - 193