Synthesis and biological activity of novel bis-indole inhibitors of bacterial transcription initiation complex formation

被引:0
|
作者
Mielczarek, Marcins [1 ]
Devakaram, Ruth V. [1 ]
Ma, Cong [2 ]
Yang, Xiao [2 ]
Kandemir, Hakan [1 ]
Purwono, Bambang [1 ]
Black, David Stc. [1 ]
Griffith, Renate [3 ]
Lewis, Peter J. [2 ]
Kumar, Naresh [1 ]
机构
[1] School of Chemistry, University of New South Wales, Sydney, NSW 2052, Australia
[2] School of Environmental and Life Sciences, University of Newcastle, Callaghan, NSW 2308, Australia
[3] School of Medical Sciences, Department of Pharmacology, University of New South Wales, Sydney, NSW 2052, Australia
来源
Organic and Biomolecular Chemistry | 2014年 / 12卷 / 18期
关键词
Anti-bacterial activity - Anti-microbial activity - Bacterial transcription - Complex formations - Gram-negative bacteria - Hydrazine hydrate - Structural feature - Structure-activity relationships;
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学科分类号
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页码:2882 / 2894
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