Synthesis of 6-Alkyl-7-oxo-4,5,6,7-tetrahydropyrazolo[1,5- c ]pyrimidine-3-carboxamides

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作者
Lombar, Klara [1 ]
Grošelj, Uroš [1 ]
Dahmann, Georg [2 ]
Stanovnik, Branko [1 ]
Svete, Jurij [1 ]
机构
[1] Faculty of Chemistry and Chemical Technology, University of Ljubljana, Večna pot 113, 1000 Ljubljana, Slovenia
[2] Boehringer Ingelheim Pharma GmbH and Co. KG, Medicinal Chemistry, Biberach,88397, Germany
关键词
Amidation - Benzyl esters - Debenzylation - histamine analogues - Methyl acrylates - Parallel synthesis - pyrazolo[1,5- c ]pyrimidines - Title compounds;
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