PHARMACOLOGICAL EFFECTS OF 2-BENZYLBENZIMIDAZOLE OPIOIDS EMERGING IN CLANDESTINE DRUG MARKETS WORLDWIDE

被引:0
|
作者
Baumann, Michael [1 ]
Walther, Donna [1 ]
Tsai, Meng-Hua [1 ]
Chen, Li [1 ]
Vandeputte, Marthe [2 ]
Stove, Christophe [2 ]
Shi, Lei [1 ]
Glatfelter, Grant [1 ]
机构
[1] NIDA, Intramural Res Program, Baltimore, MD USA
[2] Univ Ghent, Ghent, Belgium
关键词
D O I
10.1016/j.drugalcdep.2023.110070
中图分类号
R194 [卫生标准、卫生检查、医药管理];
学科分类号
摘要
引用
收藏
页数:1
相关论文
共 28 条
  • [1] Examining the mu-opioid receptor bias of fentanyl and 2-benzylbenzimidazole opioids in clandestine drug markets
    Tsai, Meng-Hua M.
    Chen, Li
    Baumann, Michael H.
    Shi, Lei
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2023, 385
  • [2] In vitro structure-activity relationships and forensic case series of emerging 2-benzylbenzimidazole 'nitazene' opioids
    De Vrieze, Liam M.
    Walton, Sara E.
    Pottie, Eline
    Papsun, Donna
    Logan, Barry K.
    Krotulski, Alex J.
    Stove, Christophe P.
    Vandeputte, Marthe M.
    ARCHIVES OF TOXICOLOGY, 2024, 98 (09) : 2999 - 3018
  • [3] When a Prophecy Comes True: Ethyleneoxynitazene as a 'Prophetic' Member of the Emerging Class of 2-Benzylbenzimidazole 'Nitazene' Synthetic Opioids
    Vandeputte, Marthe
    Glatfelter, Grant
    Walther, Donna
    Ujvary, Istvan
    Iula, Donna
    Baumann, Michael
    Stove, Christophe
    DRUG AND ALCOHOL DEPENDENCE, 2024, 260
  • [4] Pharmacological Profiling of Non-Fentanyl Synthetic Opioids That are Appearing in Clandestine Drug Markets
    Baumann, Michael
    Walther, Donna
    Glatfelter, Grant
    NEUROPSYCHOPHARMACOLOGY, 2021, 46 (SUPPL 1) : 467 - 467
  • [5] Synthesis, Chemical Characterization, and μ-Opioid Receptor Activity Assessment of the Emerging Group of "Nitazene" 2-Benzylbenzimidazole Synthetic Opioids
    Vandeputte, Marthe M.
    Van Uytfanghe, Katleen
    Layle, Nathan K.
    St Germaine, Danielle M.
    Iula, Donna M.
    Stove, Christophe P.
    ACS CHEMICAL NEUROSCIENCE, 2021, 12 (07): : 1241 - 1251
  • [6] Alkoxy chain length governs the potency of 2-benzylbenzimidazole ‘nitazene’ opioids associated with human overdose
    Grant C. Glatfelter
    Marthe M. Vandeputte
    Li Chen
    Donna Walther
    Meng-Hua M. Tsai
    Lei Shi
    Christophe P. Stove
    Michael H. Baumann
    Psychopharmacology, 2023, 240 : 2573 - 2584
  • [7] Alkoxy Chain Length Governs the In Vitro and In Vivo Potency of 2-Benzylbenzimidazole Opioids Implicated in Human Overdose Deaths
    Baumann, Michael
    Walther, Donna
    Vandeputte, Marthe M.
    Tsai, Meng-Hua M.
    Chen, Li
    Stove, Christophe P.
    Glatfelter, Grant
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2023, 385
  • [8] Alkoxy chain length governs the potency of 2-benzylbenzimidazole nitazene' opioids associated with human overdose
    Glatfelter, Grant C.
    Vandeputte, Marthe M.
    Chen, Li
    Walther, Donna
    Tsai, Meng-Hua M.
    Shi, Lei
    Stove, Christophe P.
    Baumann, Michael H.
    PSYCHOPHARMACOLOGY, 2023, 240 (12) : 2573 - 2584
  • [9] Pharmacological evaluation and forensic case series of N-pyrrolidino etonitazene (etonitazepyne), a newly emerging 2-benzylbenzimidazole ‘nitazene’ synthetic opioid
    Marthe M. Vandeputte
    Alex J. Krotulski
    Donna Walther
    Grant C. Glatfelter
    Donna Papsun
    Sara E. Walton
    Barry K. Logan
    Michael H. Baumann
    Christophe P. Stove
    Archives of Toxicology, 2022, 96 : 1845 - 1863
  • [10] Pharmacological evaluation and forensic case series of N-pyrrolidino etonitazene (etonitazepyne), a newly emerging 2-benzylbenzimidazole 'nitazene' synthetic opioid
    Vandeputte, Marthe M.
    Krotulski, Alex J.
    Walther, Donna
    Glatfelter, Grant C.
    Papsun, Donna
    Walton, Sara E.
    Logan, Barry K.
    Baumann, Michael H.
    Stove, Christophe P.
    ARCHIVES OF TOXICOLOGY, 2022, 96 (06) : 1845 - 1863