共 50 条
- [1] Mechanisms of acquired resistance to KRAS G12C inhibition in cancer.CANCER RESEARCH, 2021, 81 (13)论文数: 引用数: h-index:机构:Liu, Shengwu论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAArbour, Kathryn论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Dana Farber Canc Inst, Boston, MA 02115 USAZhu, Viola论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Irvine, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAJohnson, Melissa论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Nashville, TN USA Dana Farber Canc Inst, Boston, MA 02115 USAHeist, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Dana Farber Canc Inst, Boston, MA 02115 USAPatil, Tejas论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Aurora, CO USA Dana Farber Canc Inst, Boston, MA 02115 USARiely, Gregory论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Dana Farber Canc Inst, Boston, MA 02115 USAJacobson, Joseph论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Yang, Xiaoping论文数: 0 引用数: 0 h-index: 0机构: Broad Inst, Cambridge, MA USA Dana Farber Canc Inst, Boston, MA 02115 USAPersky, Nicole论文数: 0 引用数: 0 h-index: 0机构: Broad Inst, Cambridge, MA USA Dana Farber Canc Inst, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Sholl, Lynette论文数: 0 引用数: 0 h-index: 0机构: Brigham & Womens Hosp, 75 Francis St, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USALim, Lee论文数: 0 引用数: 0 h-index: 0机构: Resolut Biosci, Kirkland, WA USA Dana Farber Canc Inst, Boston, MA 02115 USAGarg, Kavita论文数: 0 引用数: 0 h-index: 0机构: Resolut Biosci, Kirkland, WA USA Dana Farber Canc Inst, Boston, MA 02115 USALi, Mark论文数: 0 引用数: 0 h-index: 0机构: Resolut Biosci, Kirkland, WA USA Dana Farber Canc Inst, Boston, MA 02115 USAEngstrom, Lars论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAWaters, Laura论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USALawson, J. David论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAOlson, Peter论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAChristensen, James论文数: 0 引用数: 0 h-index: 0机构: Mirati Therapeut, San Diego, CA USA Dana Farber Canc Inst, Boston, MA 02115 USALito, Piro论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY USA Dana Farber Canc Inst, Boston, MA 02115 USAOu, Sai-Hong Inatius论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Irvine, CA USA Dana Farber Canc Inst, Boston, MA 02115 USAJanne, Pasi论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USAAguirre, Andrew论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Dana Farber Canc Inst, Boston, MA 02115 USA
- [2] Multiple Mechanisms Underlie the Acquired Resistance to KRAS G12C InhibitionCANCER DISCOVERY, 2022, 12 (03)Tsai, Y. S.论文数: 0 引用数: 0 h-index: 0Woodcock, M. G.论文数: 0 引用数: 0 h-index: 0Azam, S. H.论文数: 0 引用数: 0 h-index: 0Thorne, L. B.论文数: 0 引用数: 0 h-index: 0Kanchi, K. L.论文数: 0 引用数: 0 h-index: 0Parker, J. S.论文数: 0 引用数: 0 h-index: 0
- [3] 针对KRAS G12C的首个抗肿瘤药物——AMG 510临床药物治疗杂志, 2020, 18 (05) : 31 - 34王灵智论文数: 0 引用数: 0 h-index: 0机构: 辽宁石油化工大学化学化工与环境学部 国家应急防控药物工程技术研究中心中国人民解放军军事科学院军事医学研究院 辽宁石油化工大学化学化工与环境学部于芳论文数: 0 引用数: 0 h-index: 0机构: 国家应急防控药物工程技术研究中心中国人民解放军军事科学院军事医学研究院 辽宁石油化工大学化学化工与环境学部何宇鹏论文数: 0 引用数: 0 h-index: 0机构: 辽宁石油化工大学化学化工与环境学部 辽宁石油化工大学化学化工与环境学部李行舟论文数: 0 引用数: 0 h-index: 0机构: 国家应急防控药物工程技术研究中心中国人民解放军军事科学院军事医学研究院 辽宁石油化工大学化学化工与环境学部
- [4] Mechanisms of Resistance to KRAS G12C InhibitorsJOURNAL OF THORACIC ONCOLOGY, 2021, 16 (03) : S96 - S96Ambrogio, C.论文数: 0 引用数: 0 h-index: 0机构: Univ Torino, Mol Biotechnol Ctr Mbc, Turin, Italy Univ Torino, Mol Biotechnol Ctr Mbc, Turin, Italy
- [5] The clinical KRAS(G12C) inhibitor AMG 510 drives anti-tumour immunityNATURE, 2019, 575 (7781) : 217 - +Canon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USARex, Karen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAMohr, Christopher论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USACooke, Keegan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USABagal, Dhanashri论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, San Francisco, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAGaida, Kevin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAHolt, Tyler论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAKnutson, Charles G.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Cambridge, MA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAKoppada, Neelima论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Cambridge, MA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USALanman, Brian A.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAWerner, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USARapaport, Aaron S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, San Francisco, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USASan Miguel, Tisha论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAOrtiz, Roberto论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Cambridge, MA USA Pfizer, La Jolla, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USASun, Ji-Rong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAZhu, Xiaochun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Cambridge, MA USA Takeda, Cambridge, MA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAMcCarter, John D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAVolak, Laurie P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Cambridge, MA USA Celgene, San Diego, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAHouk, Brett E.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Clin Dev, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAFakih, Marwan G.论文数: 0 引用数: 0 h-index: 0机构: City Hope Natl Med Ctr, Duarte, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAO'Neil, Bert H.论文数: 0 引用数: 0 h-index: 0机构: Indiana Univ Sch Med, Indianapolis, IN 46202 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAPrice, Timothy J.论文数: 0 引用数: 0 h-index: 0机构: Queen Elizabeth Hosp, Woodville, SA, Australia Univ Adelaide, Adelaide, SA, Australia Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAFalchook, Gerald S.论文数: 0 引用数: 0 h-index: 0机构: Sarah Cannon Res Inst, Denver, CO USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USADesai, Jayesh论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Canc Ctr, Melbourne, Vic, Australia Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAKuo, James论文数: 0 引用数: 0 h-index: 0机构: Scientia Clin Res, Randwick, NSW, Australia Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA论文数: 引用数: h-index:机构:Hong, David S.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAOuyang, Wenjun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, San Francisco, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAHenary, Haby论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Clin Dev, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USAArvedson, Tara论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, San Francisco, CA USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USACee, Victor J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USALipford, J. Russell论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA Amgen Inc, Amgen Res, Thousand Oaks, CA 91320 USA
- [6] The clinical KRAS(G12C) inhibitor AMG 510 drives anti-tumour immunityNature, 2019, 575 : 217 - 223Jude Canon论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchKaren Rex论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchAnne Y. Saiki论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchChristopher Mohr论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchKeegan Cooke论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchDhanashri Bagal论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchKevin Gaida论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchTyler Holt论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchCharles G. Knutson论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchNeelima Koppada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchBrian A. Lanman论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchJonathan Werner论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchAaron S. Rapaport论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchTisha San Miguel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchRoberto Ortiz论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchTao Osgood论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchJi-Rong Sun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchXiaochun Zhu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchJohn D. McCarter论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchLaurie P. Volak论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchBrett E. Houk论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchMarwan G. Fakih论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchBert H. O’Neil论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchTimothy J. Price论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchGerald S. Falchook论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchJayesh Desai论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchJames Kuo论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchRamaswamy Govindan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchDavid S. Hong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchWenjun Ouyang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchHaby Henary论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchTara Arvedson论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchVictor J. Cee论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen ResearchJ. Russell Lipford论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc,Amgen Research
- [7] EMT is a cause of both intrinsic and acquired resistance to KRAS G12C inhibitor in KRAS G12C mutant NSCLCANNALS OF ONCOLOGY, 2021, 32 : S307 - S307Adachi, Yuta论文数: 0 引用数: 0 h-index: 0机构: Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, Japan Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, JapanIto, Kentaro论文数: 0 引用数: 0 h-index: 0机构: Matsusaka City Hosp, Dept Resp Med, Matsusaka, Mie, Japan Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, JapanKimura, Ryo论文数: 0 引用数: 0 h-index: 0机构: Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, Japan Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, JapanYamaguchi, Rui论文数: 0 引用数: 0 h-index: 0机构: Aichi Canc Ctr, Res Inst, Div Canc Syst Biol, Nagoya, Aichi, Japan Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, JapanEbi, Hiromichi论文数: 0 引用数: 0 h-index: 0机构: Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, Japan Aichi Canc Ctr, Res Inst, Div Mol Therapeut, Nagoya, Aichi, Japan
- [8] Targeting KRAS G12C mutations in colorectal cancerGASTROENTEROLOGY REPORT, 2023, 11Zhao, Ming-He论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Key Lab Carcinogenesis & Translat Res, Minist Educ, Canc Hosp & Inst,Unit 3,Gastrointestinal Canc Ctr, 52 Fucheng Rd, Beijing 100142, Peoples R China Peking Univ, Key Lab Carcinogenesis & Translat Res, Minist Educ, Canc Hosp & Inst,Unit 3,Gastrointestinal Canc Ctr, 52 Fucheng Rd, Beijing 100142, Peoples R ChinaWu, Ai-Wen论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Key Lab Carcinogenesis & Translat Res, Minist Educ, Canc Hosp & Inst,Unit 3,Gastrointestinal Canc Ctr, 52 Fucheng Rd, Beijing 100142, Peoples R China Peking Univ, Key Lab Carcinogenesis & Translat Res, Minist Educ, Canc Hosp & Inst,Unit 3,Gastrointestinal Canc Ctr, 52 Fucheng Rd, Beijing 100142, Peoples R China
- [9] CodeBreaK 200: Sotorasib (AMG510) Has Broken the KRAS G12C+ NSCLC Enigma CodeLUNG CANCER-TARGETS AND THERAPY, 2023, 14 : 31 - 39Brazel, Danielle论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Internal Med, Div Hematol Oncol, Sch Med, Orange, CA USA Univ Calif Irvine, Dept Internal Med, Div Hematol Oncol, Sch Med, Orange, CA USAKim, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Internal Med, Div Hematol Oncol, Sch Med, Orange, CA USA Univ Calif Irvine, Dept Internal Med, Div Hematol Oncol, Sch Med, Orange, CA USAOu, Sai-Hong Ignatius论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Irvine, Dept Internal Med, Div Hematol Oncol, Sch Med, Orange, CA USA Chao Family Comprehens Canc Ctr, Orange, CA USA Univ Calif Irvine, Chao Family Comprehens Canc Ctr, Dept Med, Div Hematol Med Oncol,Sch Med, 200 South Manchester Ave,Suite 400, Orange, CA 92868 USA Univ Calif Irvine, Dept Internal Med, Div Hematol Oncol, Sch Med, Orange, CA USA
- [10] KRAS G12C Mutations in NSCLC: From Target to ResistanceCANCERS, 2021, 13 (11)论文数: 引用数: h-index:机构:Banna, Giuseppe Luigi论文数: 0 引用数: 0 h-index: 0机构: Portsmouth Hosp NHS Trust, Dept Oncol, Portsmouth PO2 8QD, England Switzerland Univ Geneva, Univ Hosp Geneva, Dept Oncol, Swiss Canc Ctr Leman, CH-1205 Geneva, Switzerland论文数: 引用数: h-index:机构: