MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY OF DIACYLGLYCEROL LIPASE AND KINASE INHIBITORS

被引：5
|
作者：
SEKAR, MC [1 ]
DICKINSON, KEJ [1 ]
PRUITT, RE [1 ]
HIRSCHOWITZ, BI [1 ]
HOKIN, LE [1 ]
机构：
[1] UNIV ALABAMA,DIV GASTROENTEROL,BIRMINGHAM,AL 35294
来源：
BIOCHEMICAL PHARMACOLOGY | 1990年 / 39卷 / 12期
关键词：
D O I：
10.1016/0006-2952(90)90634-W
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
[No abstract available]
引用
收藏
页码：2069 / 2073
页数：5
相关论文
共 50 条
  • [1] THE ROLE OF DIACYLGLYCEROL IN THE EXOCYTOSIS OF THE SPERM ACROSOME - STUDIES USING DIACYLGLYCEROL LIPASE AND DIACYLGLYCEROL KINASE INHIBITORS AND EXOGENOUS DIACYLGLYCEROLS
    ROLDAN, ERS
    HARRISON, RAP
    BIOCHEMICAL JOURNAL, 1992, 281 : 767 - 773
  • [2] THE ACTIONS OF INHIBITORS OF DIACYLGLYCEROL KINASE AND DIACYLGLYCEROL LIPASE ON HISTAMINE-RELEASE FROM RAT PERITONEAL MAST-CELLS
    CANTWELL, ME
    FOREMAN, JC
    BRITISH JOURNAL OF PHARMACOLOGY, 1987, 92 (03) : 597 - 601
  • [3] INHIBITORS OF DIACYLGLYCEROL LIPASE AND DIACYLGLYCEROL KINASE INHIBIT CARBAMYLCHOLINE-STIMULATED RESPONSES IN GUINEA-PIG PANCREATIC MINILOBULES
    SEKAR, MC
    HOKIN, LE
    ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS, 1987, 256 (02) : 509 - 514
  • [4] BENZOQUINOID TYROSINE KINASE INHIBITORS BLOCK MUSCARINIC RECEPTOR FUNCTION
    OTERO, AD
    SWEITZER, NM
    FASEB JOURNAL, 1993, 7 (07): : A1159 - A1159
  • [5] Assay and inhibition of diacylglycerol lipase activity
    Johnston, Meghan
    Bhatt, Shachi R.
    Sikka, Surina
    Mercier, Richard W.
    West, Jay M.
    Makriyannis, Alexandros
    Gatley, S. John
    Duclos, Richard I., Jr.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (14) : 4585 - 4592
  • [6] INFLUENCE OF PHORBOL ESTERS, AND DIACYLGLYCEROL KINASE AND LIPASE INHIBITORS ON NORADRENALINE RELEASE AND PHOSPHOINOSITIDE HYDROLYSIS IN CHROMAFFIN CELLS
    JONES, JA
    OWEN, PJ
    BOARDER, MR
    BRITISH JOURNAL OF PHARMACOLOGY, 1990, 101 (03) : 521 - 526
  • [7] Endocannabinoids and diacylglycerol kinase activity
    Gantayet, Arpita
    Jegatheswaran, Januvi
    Jayakumaran, Gowtham
    Topham, Matthew K.
    Epand, Richard M.
    BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES, 2011, 1808 (04): : 1050 - 1053
  • [8] ISOMERIZATION OF THE MUSCARINIC RECEPTOR - ANTAGONIST COMPLEX
    JARV, J
    HEDLUND, B
    BARTFAI, T
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1979, 254 (13) : 5595 - 5598
  • [9] BENZOQUINOID TYROSINE KINASE INHIBITORS ARE POTENT BLOCKERS OF CARDIAC MUSCARINIC RECEPTOR FUNCTION
    OTERO, AD
    SWEITZER, NM
    MOLECULAR PHARMACOLOGY, 1993, 44 (03) : 595 - 604
  • [10] Comprehensive Analysis of Structure-Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α Inhibitors
    Janssen, Freek J.
    Baggelaar, Marc P.
    Hummel, Jessica J. A.
    Overkleeft, Herman S.
    Cravatt, Benjamin F.
    Boger, Dale L.
    van der Stelt, Mario
    JOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (24) : 9742 - 9753
12345