AVERMECTIN-MILBEMYCIN SYNTHETIC STUDIES .6. STEREOSELECTIVE ELABORATION OF THE SOUTHERN-HEMISPHERE OXAHYDRINDENE

被引：9

作者：

FUJIWARA, S

SMITH, AB

机构：

[1] UNIV PENN,DEPT CHEM,RES STRUCT MATTER LAB,PHILADELPHIA,PA 19104

[2] UNIV PENN,MONELL CHEM SENSES CTR,PHILADELPHIA,PA 19104

来源：

TETRAHEDRON LETTERS | 1992年 / 33卷 / 09期

基金：

美国国家卫生研究院;

关键词：

D O I：

10.1016/S0040-4039(00)91891-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An economic, stereoselective synthesis of the highly oxygenated oxahydrindene nucleus of the avermectin-milbemycin family of anthelmintics has been achieved, exploiting a facile intramolecular S(N)2' cyclization as the key step.

引用

页码：1185 / 1188

页数：4

共 8 条

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