SYNTHESIS OF IMIDAZOBENZAZEPINTHIONES - A NEW SERIES OF HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS

被引：8
|
作者：
SALASKI, EJ
机构：
来源：
TETRAHEDRON LETTERS | 1995年 / 36卷 / 09期
关键词：
D O I：
10.1016/0040-4039(95)00006-X
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A general route to a series of novel imidazobenzazepines that are ''carba'' analogs of the TIBO class of non-nucleoside HIV-1 reverse transcriptase inhibitors has been developed. A pair of allyl side-chain containing compounds were found to have significant HIV-1 inhibitory activity.
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页码：1387 / 1390
页数：4
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