RELATIVE ACTIVITIES OF SCH 23390 AND ITS ANALOGS IN 3 TESTS FOR D1/DA1 DOPAMINE RECEPTOR ANTAGONISM

被引:38
|
作者
BARNETT, A
AHN, H
BILLARD, W
GOLD, EH
KOHLI, JD
GLOCK, D
GOLDBERG, LI
机构
[1] UNIV CHICAGO, DEPT PHARMACOL & PHYSIOL SCI,COMM CLIN PHARMACOL, CHICAGO, IL 60637 USA
[2] UNIV CHICAGO, DEPT MED,COMM CLIN PHARMACOL, CHICAGO, IL 60637 USA
关键词
D O I
10.1016/0014-2999(86)90772-7
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:249 / 253
页数:5
相关论文
共 50 条
  • [1] SYNTHESIS OF A RADIOBROMINATED ANALOG OF SCH-23390, A SELECTIVE DOPAMINE D1/DA1 ANTAGONIST
    DEJESUS, OT
    VANMOFFAERT, GJ
    GLOCK, D
    GOLDBERG, LI
    FRIEDMAN, AM
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1986, 23 (09): : 919 - 925
  • [2] POSITRON TOMOGRAPHY OF A RADIO-BROMINATED ANALOG OF THE D1/DA1 ANTAGONIST, SCH-23390
    FRIEDMAN, AM
    DEJESUS, OT
    WOOLVERTON, WL
    VANMOFFAERT, G
    GOLDBERG, LI
    PRASAD, A
    BARNETT, A
    DINERSTEIN, RJ
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1985, 108 (03) : 327 - 328
  • [3] In Vivo DA D1 Receptor Selectivity of NNC 112 and SCH 23390
    Jesper Ekelund
    Mark Slifstein
    Raj Narendran
    Olivier Guillin
    Hemant Belani
    Ning-Ning Guo
    Yuying Hwang
    Dah-Ren Hwang
    Anissa Abi-Dargham
    Marc Laruelle
    Molecular Imaging and Biology, 2007, 9
  • [4] BLOCKADE OF RENAL EFFECTS OF DOPAMINE IN THE DOG BY THE DA1 ANTAGONIST SCH-23390
    FREDERICKSON, ED
    BRADLEY, T
    GOLDBERG, LI
    AMERICAN JOURNAL OF PHYSIOLOGY, 1985, 249 (02): : F236 - F240
  • [5] In vivo DA D1 receptor selectivity of NNC 112 and SCH 23390
    Ekelund, Jesper
    Slifstein, Mark
    Narendran, Raj
    Guillin, Olivier
    Belani, Hemant
    Guo, Ning-Ning
    Hwang, Yuying
    Hwang, Dah-Ren
    Abi-Dargham, Anissa
    Laruelle, Marc
    MOLECULAR IMAGING AND BIOLOGY, 2007, 9 (03) : 117 - 125
  • [6] POSITRON-EMITTING ANALOGS OF SCH 23390 FOR THE STUDY OF DOPAMINE D1 RECEPTORS
    DEJESUS, OT
    WOOLVERTON, WL
    VANMOFFAERT, GJC
    COOPER, MD
    FRIEDMAN, AM
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1986, 23 (10-12): : 1403 - 1404
  • [7] SEPARATION OF PERIPHERAL DOPAMINE-RECEPTORS BY A SELECTIVE DA1 ANTAGONIST, SCH-23390
    GOLDBERG, LI
    GLOCK, D
    KOHLI, JD
    BARNETT, A
    HYPERTENSION, 1984, 6 (02) : I25 - I30
  • [8] AUTORADIOGRAPHIC LOCALIZATION OF DOPAMINE DA1 RECEPTORS IN RAT-KIDNEY WITH [H-3]SCH 23390
    HUO, T
    HEALY, DP
    AMERICAN JOURNAL OF PHYSIOLOGY, 1989, 257 (03): : F414 - F423
  • [9] SYNTHESIS OF [C-11] SCH 23390 FOR DOPAMINE D1 RECEPTOR STUDIES
    DEJESUS, OT
    VANMOFFAERT, GJC
    FRIEDMAN, AM
    APPLIED RADIATION AND ISOTOPES, 1987, 38 (05) : 345 - 348
  • [10] Binding of [3H]SCH23390 to Dopamine D1 receptor synthesized with liposomes
    Arimitsu, Eiji
    Ogasawara, Tomio
    Hiasa, Yoich
    Onji, Morikazu
    Sawazaki, Tatsuya
    Maeyama, Kazutaka
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2013, 121 : 127P - 127P