BETA-CARBOLINE ALKALOIDS .8. REGIOSELECTIVE HOMOLYTIC ACETYLATION OF BETA-CARBOLINES

被引：14
|
作者：
BRACHER, F
DAAB, J
机构：
[1] Institut für Pharmazeutische Chemie, Technische Universität Braunschweig, D-38106 Braunschweig
来源：
SYNTHETIC COMMUNICATIONS | 1995年 / 25卷 / 10期
关键词：
D O I：
10.1080/00397919508011768
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Homolytic acetylation of 3-ethoxycarbonyl-beta-carboline and norharmane occurs selectively at 1-position. Better yields are obtained by generation of the acetyl radical from acetaldehyde than by oxidative decarboxylation of pyruvic acid.
引用
收藏
页码：1557 / 1562
页数：6
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