INTERACTION OF THE ANTIOESTROGEN ICI-164,384 WITH THE ESTROGEN-RECEPTOR

被引:78
|
作者
WEATHERILL, PJ [1 ]
WILSON, APM [1 ]
NICHOLSON, RI [1 ]
DAVIES, P [1 ]
WAKELING, AE [1 ]
机构
[1] ICI PLC,DIV PHARMACEUT,ALDERLEY PK,CHESHIRE,ENGLAND
关键词
D O I
10.1016/0022-4731(88)90103-3
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:263 / 266
页数:4
相关论文
共 50 条
  • [1] ANTIESTROGEN ICI-164,384 REDUCES CELLULAR ESTROGEN-RECEPTOR CONTENT BY INCREASING ITS TURNOVER
    DAUVOIS, S
    DANIELIAN, PS
    WHITE, R
    PARKER, MG
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1992, 89 (09) : 4037 - 4041
  • [2] EFFECTS OF THE ANTIOESTROGEN, ICI-164,384, ON ESTROGEN-INDUCED RNAS IN MCF-7 CELLS
    WISEMAN, LR
    WAKELING, AE
    MAY, FEB
    WESTLEY, BR
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1989, 33 (01): : 1 - 6
  • [3] THE MECHANISM OF ICI-164,384 ANTIESTROGENICITY INVOLVES RAPID LOSS OF ESTROGEN-RECEPTOR IN UTERINE TISSUE
    GIBSON, MK
    NEMMERS, LA
    BECKMAN, WC
    DAVIS, VL
    CURTIS, SW
    KORACH, KS
    ENDOCRINOLOGY, 1991, 129 (04) : 2000 - 2010
  • [4] EFFECTS OF THE ANTIOESTROGEN ICI-164,384 ON ESTROGEN-INDUCED RNAS IN MCF-7 CELLS
    WISEMAN, LR
    WAKELING, AE
    MAY, FEB
    WESTLEY, BR
    BIOCHEMICAL SOCIETY TRANSACTIONS, 1988, 16 (06) : 1063 - 1063
  • [5] INHIBITION OF ESTROGEN-RECEPTOR DNA-BINDING BY THE PURE ANTIESTROGEN ICI-164,384 APPEARS TO BE MEDIATED BY IMPAIRED RECEPTOR DIMERIZATION
    FAWELL, SE
    WHITE, R
    HOARE, S
    SYDENHAM, M
    PAGE, M
    PARKER, MG
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1990, 87 (17) : 6883 - 6887
  • [6] INHIBITION OF NUCLEAR TRANSPORT IS NOT ESSENTIAL FOR INHIBITION OF RECEPTOR FUNCTION BY THE TYPE-II ESTROGEN ANTAGONIST ICI-164,384
    MIKSICEK, RJ
    LEE, C
    TOPPRAPIEJKO, K
    NEFF, S
    STEROID RECEPTORS AND ANTIHORMONES, 1995, 761 : 361 - 364
  • [7] A COMPARATIVE-STUDY OF THE INTERACTION OF ESTRADIOL AND THE STEROIDAL PURE ANTIESTROGEN, ICI 164,384, WITH THE MOLYBDATE-STABILIZED ESTROGEN-RECEPTOR
    WILSON, APM
    WEATHERILL, PJ
    NICHOLSON, RI
    DAVIES, P
    WAKELING, AE
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1990, 35 (3-4): : 421 - 428
  • [8] ICI-164,384, A PURE ANTAGONIST OF ESTROGEN-STIMULATED MCF-7 CELL-PROLIFERATION AND INVASIVENESS
    THOMPSON, EW
    KATZ, D
    SHIMA, TB
    WAKELING, AE
    LIPPMAN, ME
    DICKSON, RB
    CANCER RESEARCH, 1989, 49 (24) : 6929 - 6934
  • [9] ANTAGONISM OF ESTROGEN-INDUCED AND ANTIESTROGEN-INDUCED UTERINE COMPLEMENT COMPONENT C3 EXPRESSION BY ICI-164,384
    GALMAN, MS
    SUNDSTROM, SA
    LYTTLE, CR
    JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1990, 36 (04): : 281 - 286
  • [10] STUDIES ON THE ACTIVATION OF THE ESTROGEN-RECEPTOR BOUND TO THE ANTIESTROGENS 4-HYDROXYTAMOXIFEN AND ICI 164,384 BY USING 3 MONOCLONAL-ANTIBODIES
    GIAMBIAGI, N
    PASQUALINI, JR
    JOURNAL OF MOLECULAR ENDOCRINOLOGY, 1991, 7 (01) : 9 - 19