INHIBITION AND REVERSAL OF METHOTREXATE-H-3 (MTX) BINDING TO DIHYDROFOLATE-REDUCTASE (DHFR) BY DIHYDROFOLATE (H2F) - RELATIONSHIP TO INTRACELLULAR (IC) EVENTS

被引：0

作者：

WHITE, JC ^{[1
]}

GOLDMAN, ID ^{[1
]}

机构：

[1] MED COLL VIRGINIA,RICHMOND,VA 23298

来源：

PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH | 1979年 / 20卷 / MAR期

关键词：

D O I：

暂无

中图分类号：

R73 [肿瘤学];

学科分类号：

100214 ;

摘要：

引用

页码：263 / 263

页数：1

共 17 条

[1] RELATIVE POTENCY OF INHIBITION OF DIHYDROFOLATE-REDUCTASE (DHFR) BY INTRACELLULAR FOLATES AND BY METHOTREXATE (MTX) AND ITS METABOLITES
DRAKE, JC
ALLEGRA, CJ
GOLDMAN, ID
KAUFMAN, B
BARAM, J
CHABNER, BA
PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1986, 27 : 257 - 257
[2] QUANTITATIVE ASPECTS OF METHOTREXATE (MTX) BINDING BY L-1210 DIHYDROFOLATE-REDUCTASE (DHFR)
ROTHENBERG, SP
DACOSTA, M
IQBAL, MP
PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1976, 17 (MAR): : 106 - 106
[3] AUGMENTATION OF H-3-METHOTREXATE (MTX) BINDING TO DIHYDROFOLATE-REDUCTASE (DHFR) BY SULFAMETHOXAZOLE (SM) - EVIDENCE FOR SIMULTANEOUS BINDING OF 2 INHIBITORS AT PTEROATE BINDING-SITE
WHITE, JC
GOLDMAN, ID
FEDERATION PROCEEDINGS, 1976, 35 (07) : 1572 - 1572
[4] ASSESSMENT OF DIHYDROFOLATE REDUCTASE (H2FR) ACTIVITY IN-VIVO AFTER ADMINISTRATION OF H-3-DIHYDROFOLATE (H2F)
MISHRA, LC
PARMAR, AS
MEAD, JAR
PHARMACOLOGIST, 1971, 13 (02): : 208 - &
[5] RAPID ANALYSIS OF THE CONSEQUENCES OF DIHYDROFOLATE-REDUCTASE (DHFR) INHIBITION BY METHOTREXATE (MTX) OR TRIMETREXATE (TMQ) IN L1210 CELLS
SEITHER, RL
GOLDMAN, ID
PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1988, 29 : 282 - 282
[6] DIHYDROFOLATE-REDUCTASE (DHFR) FROM A METHOTREXATE-RESISTANT HUMAN-BREAST CANCER CELL-LINE - PURIFICATION, PROPERTIES, AND BINDING OF METHOTREXATE (MTX) AND POLYGLUTAMATES
CLENDENINN, NJ
COWAN, KH
KAUFMAN, BT
NADKARNI, MV
CHABNER, BA
PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1983, 24 (MAR): : 276 - 276
[7] CELL-DENSITY DEPENDENT INHIBITION OF 7-HYDROXY (7-OH) METHOTREXATE (MTX) AT THE LEVEL OF DIHYDROFOLATE-REDUCTASE (DHFR) AND AICAR TRANSFORMYLASE (AT)
SEITHER, RL
GOLDMAN, ID
PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1987, 28 : 274 - 274
[8] PTERIN 1H-3H TAUTOMERISM AND ITS POSSIBLE RELEVANCE TO THE BINDING OF FOLATE TO DIHYDROFOLATE-REDUCTASE
SCHWALBE, CH
LOWIS, DR
RICHARDS, WG
JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS, 1993, (15) : 1199 - 1200
[9] A H-1-NMR STUDY OF THE ROLE OF THE GLUTAMATE MOIETY IN THE BINDING OF METHOTREXATE TO LACTOBACILLUS-CASEI DIHYDROFOLATE-REDUCTASE
ANTONJUK, DJ
BIRDSALL, B
CHEUNG, HTA
CLORE, GM
FEENEY, J
GRONENBORN, A
ROBERTS, GCK
TRAN, TQ
BRITISH JOURNAL OF PHARMACOLOGY, 1984, 81 (02) : 309 - 315
[10] INHIBITION OF HUMAN DIHYDROFOLATE-REDUCTASE (DHFR) BY POLYGLUTAMYL DERIVATIVES OF METHOTREXATE (MTX), 10-DEAZAAMINOPTERIN (10-DAM) AND 10-ETHYL-10-DE-AZAAMINOPTERIN (10-EDAM)
KUMAR, P
GAUMONT, Y
KISLIUK, RL
FREISHEIM, JH
NAIR, MG
PROCEEDINGS OF THE AMERICAN ASSOCIATION FOR CANCER RESEARCH, 1987, 28 : 274 - 274

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