ON THE SYNTHESIS OF PHOSPHONAMIDATE PEPTIDES

被引：35

作者：

MUSIOL, HJ ^{[1
]}

GRAMS, F ^{[1
]}

RUDOLPHBOHNER, S ^{[1
]}

MORODER, L ^{[1
]}

机构：

[1] MAX PLANCK INST BIOCHEM,D-82152 MARTINSRIED,GERMANY

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1994年 / 59卷 / 21期

关键词：

D O I：

10.1021/jo00100a007

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Oxalyl chloride-mediated preparation of phosphonochloridates allowed the improvement of the synthesis of phosphonamidate peptides, particularly if AgCN was used as catalyst or upon conversion of the chloridate into the 7-aza-1-hydroxybenzotriazole ester.

引用

页码：6144 / 6146

页数：3

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