Structure-activity relationships of quinone and acridone photosystem II inhibitors

被引:0
|
作者
Draber, W [1 ]
Trebst, A [1 ]
Oettmeier, W [1 ]
机构
[1] RUHR UNIV BOCHUM, LEHRSTUHL BIOCHEM PFLANZEN, D-44780 BOCHUM, GERMANY
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中图分类号
S3 [农学(农艺学)];
学科分类号
0901 ;
摘要
Photosynthesis inhibition was determined with thylakoids of the green alga Chlamydomonas reinhardtii on eleven acridones, twelve 1,4-benzoquinones and fifteen 1,4-naphthoquinones. The wild type and five mutants of the algae were used. The mutants had known changes in the inhibitor-binding region of the D-1 protein. The compounds showed reduced as well as enhanced inhibitory activity up to two orders of magnitude. Their resistance/supersensitivity pattern and structure-activity studies revealed that the inhibitory behaviour resembles that of the nitrophenols.
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页码:186 / 198
页数:13
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